SCHEMBL7053088

SCHEMBL7053088

O=C(NCCCCN1CCC(Nc2cccc(C(F)(F)F)c2)CC1)c1ccc(-c2cn3ccsc3n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 6/20 0.49
DRD2 P14416 5/20 0.49
ADRA1A P35348 1/20 0.45
DRD4 P21917 2/20 0.44
TP53 P04637 3/20 0.43
PKM P14618 2/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CCR3 P51677 1/20 0.41
HTR2A P28223 1/20 0.41
CHRM4 P08173 1/20 0.40
HPGD P15428 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
UBE2M P61081 1/20 0.40
DCUN1D1 Q96GG9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7058078 0.88 DRD2 (0.56) DRD3DRD2ADRA1ADRD4RAB9A
SCHEMBL7051851 0.88 DRD3 (0.49) DRD3DRD2DRD4TP53PKM
SCHEMBL7053551 0.87 DRD2 (0.45) DRD3DRD2ADRA1ATP53ALDH1A1
SCHEMBL7115347 0.86 DRD3 (0.49) DRD3DRD2ADRA1ADRD4TP53
Hydrochloric Acid SCHEMBL7059854 0.86 CCR3 (0.51) DRD3DRD2ADRA1ADRD4CCR3
SCHEMBL7056847 0.83 DRD2 (0.49) DRD3DRD2ADRA1ADRD4TP53
SCHEMBL7119593 0.82 CCR3 (0.55) DRD3DRD2ADRA1ACCR3UBE2M
SCHEMBL7060979 0.81 DRD2 (0.52) DRD3DRD2ADRA1ADRD4CCR3
SCHEMBL7055659 0.81 DRD2 (0.50) DRD3DRD2ADRA1ACCR3UBE2M
SCHEMBL7118079 0.81 DRD2 (0.46) DRD3DRD2DRD4TP53PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028725-A1 4-(1-PIPERIDINY)-BUTYLCARBOXAMIDE AS D3 DOPAMINE RECEPTOR SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed