SCHEMBL7053551

SCHEMBL7053551

O=C(NCCCCN1CCC(Nc2cccc(C(F)(F)F)c2)CC1)c1ccc(-c2cn3cccnc3n2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.45
DRD3 P35462 9/20 0.45
ADRA1A P35348 1/20 0.44
MAPT P10636 3/20 0.42
TP53 P04637 2/20 0.42
HTR1A P08908 2/20 0.41
HTR2A P28223 2/20 0.41
HTR2C P28335 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GAA P10253 3/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
USP2 O75604 1/20 0.40
ESR1 P03372 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
NPC1 O15118 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7058078 0.89 DRD2 (0.56) DRD2DRD3ADRA1AHTR1AHTR2A
SCHEMBL7057687 0.87 CCR3 (0.50) DRD2DRD3ADRA1ACCR3
SCHEMBL7053088 0.87 DRD3 (0.49) DRD2DRD3ADRA1ATP53HTR2A
SCHEMBL7055659 0.82 DRD2 (0.50) DRD2DRD3ADRA1ACCR3
SCHEMBL7119593 0.81 CCR3 (0.55) DRD2DRD3ADRA1ACCR3
SCHEMBL7060979 0.80 DRD2 (0.52) DRD2DRD3ADRA1ACCR3
SCHEMBL7057584 0.79 DRD3 (0.69) DRD2DRD3ADRA1A
SCHEMBL7054406 0.77 DRD3 (0.57) DRD2DRD3ADRA1AHTR1AHTR2A
SCHEMBL7055557 0.76 DRD3 (0.58) DRD2DRD3ADRA1AHTR1AHTR2A
SCHEMBL7052427 0.76 DRD2 (0.48) DRD2DRD3ADRA1AHTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028725-A1 4-(1-PIPERIDINY)-BUTYLCARBOXAMIDE AS D3 DOPAMINE RECEPTOR SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed