SCHEMBL7053767

SCHEMBL7053767

CCCc1nc(N2CCN(C(CC(C)=O)On3nnc4ccccc43)CC2)c2cc(CC)sc2n1

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 17/20 0.38
MEN1 O00255 2/20 0.37
HTR6 P50406 1/20 0.36
NTSR1 P30989 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7052654 0.88 P2RY12 (0.43) P2RY12MEN1
SCHEMBL7051730 0.88 P2RY12 (0.38) P2RY12MEN1HTR6NTSR1KMT2A
SCHEMBL7052594 0.86 MEN1 (0.53) P2RY12MEN1ALDH1A1KMT2A
SCHEMBL7049798 0.80 MEN1 (0.47) P2RY12MEN1ALDH1A1KMT2A
SCHEMBL5848957 0.79 P2RY12 (0.46) P2RY12MEN1ALDH1A1KMT2A
SCHEMBL7049255 0.78 P2RY12 (0.39) P2RY12MEN1HTR6KMT2A
SCHEMBL7053983 0.78 HTR6 (0.47) P2RY12MEN1HTR6ALDH1A1KMT2A
SCHEMBL7051550 0.77 P2RY12 (0.39) P2RY12MEN1HTR6KMT2A
SCHEMBL7050548 0.77 P2RY12 (0.39) P2RY12MEN1HTR6KMT2A
SCHEMBL7052962 0.76 KMT2A (0.40) MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003022214-A2 PIPERAZINE AND HOMOPIPERAZINE COMPOUNDS MILLENNIUM PHARMACEUTICALS, INC. (US) 2003-03-20 WO disclosed