SCHEMBL7054947

SCHEMBL7054947

COc1ccccc1-c1ccc(N2CCN(CCCC#N)CC2)c(OC)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 5/20 0.53
DRD3 P35462 7/20 0.52
DRD2 P14416 6/20 0.52
HTR1A P08908 3/20 0.51
ALDH1A1 P00352 2/20 0.51
MEN1 O00255 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
ALOX12 P18054 1/20 0.51
ADRA1D P25100 1/20 0.51
ADRA1A P35348 1/20 0.51
ADRA1B P35368 1/20 0.51
KMT2A Q03164 1/20 0.51
HIF1A Q16665 1/20 0.51
HSD17B10 Q99714 1/20 0.51
KDM4E B2RXH2 1/20 0.50
GLA P06280 1/20 0.50
HPGD P15428 1/20 0.50
DRD5 P21918 2/20 0.49
DRD4 P21917 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7057457 0.89 DRD3 (0.54) DRD3DRD2HTR1ADRD4
SCHEMBL948083 0.85 DRD2 (0.71) HTR7DRD3DRD2HTR1AALDH1A1
SCHEMBL30080790 0.85 DRD2 (0.71) HTR7DRD3DRD2HTR1AALDH1A1
SCHEMBL7056834 0.84 HTR1A (0.56) HTR7DRD3DRD2HTR1AALDH1A1
SCHEMBL6954563 0.81 HTR1A (0.71) HTR7DRD3DRD2HTR1AALDH1A1
SCHEMBL27678005 0.78 DRD2 (0.54) HTR7DRD3DRD2HTR1AMEN1
SCHEMBL7057411 0.78 HTR1A (0.49) HTR7DRD3DRD2HTR1AALDH1A1
SCHEMBL6246397 0.77 DRD2 (0.69) HTR7DRD3DRD2HTR1AMEN1
SCHEMBL7054984 0.74 HTR7 (0.68) HTR7DRD3DRD2HTR1AALDH1A1
SCHEMBL7053849 0.73 DRD3 (0.56) DRD3DRD2HTR1ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028728-A1 4-(4-SUBSTITUTED PIPERAZINYL-1YL)-BUTYLCARBOXAMIDES AS D3 DOPAMINE SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed