SCHEMBL7056570

SCHEMBL7056570

COc1ccccc1NC1CCN(CCCCN2C(=O)c3ccccc3C2=O)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 1.00
ALDH1A1 P00352 2/20 0.60
HTR1A P08908 2/20 0.60
HTR7 P34969 2/20 0.60
MEN1 O00255 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
ALOX12 P18054 1/20 0.60
ADRA1D P25100 1/20 0.60
ADRA1A P35348 1/20 0.60
ADRA1B P35368 1/20 0.60
KMT2A Q03164 1/20 0.60
HIF1A Q16665 1/20 0.60
HSD17B10 Q99714 1/20 0.60
KDM4E B2RXH2 1/20 0.59
GLA P06280 1/20 0.59
HPGD P15428 1/20 0.59
HTR4 Q13639 2/20 0.58
DRD3 P35462 4/20 0.57
HTR2A P28223 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6710759 0.81 DRD2 (0.67) DRD2ALDH1A1HTR1AHTR7MEN1
SCHEMBL8042421 0.77 DRD2 (0.63) DRD2ALDH1A1HTR1AHTR7MEN1
SCHEMBL8042425 0.77 DRD2 (0.63) DRD2ALDH1A1HTR1AHTR7MEN1
SCHEMBL1463650 0.77 DRD2 (0.62) DRD2ALDH1A1HTR1AHTR7MEN1
SCHEMBL7057313 0.77 DRD2 (0.62) DRD2HTR4
SCHEMBL14761599 0.77 HTR1A (0.98) DRD2ALDH1A1HTR1AHTR7MEN1
Nan-190 SCHEMBL29389115 0.75 HTR1A (1.00) DRD2ALDH1A1HTR1AHTR7MEN1
Nan-190 SCHEMBL30080779 0.75 HTR1A (1.00) DRD2ALDH1A1HTR1AHTR7MEN1
Nan-190 SCHEMBL2231820 0.75 HTR1A (1.00) DRD2ALDH1A1HTR1AHTR7MEN1
SCHEMBL7051610 0.75 DRD2 (0.60) DRD2ALDH1A1HTR1AHTR7DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028725-A1 4-(1-PIPERIDINY)-BUTYLCARBOXAMIDE AS D3 DOPAMINE RECEPTOR SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed