SCHEMBL7057485

SCHEMBL7057485

CNC(=O)Nc1cc(-c2ccc(OC)cc2)sc1C(=O)NC

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 7/20 0.63
PTPN1 P18031 2/20 0.60
HPGD P15428 4/20 0.56
ALDH1A1 P00352 3/20 0.56
KDM4E B2RXH2 3/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
MAPT P10636 3/20 0.56
GLA P06280 2/20 0.56
GAA P10253 2/20 0.56
NPC1 O15118 1/20 0.56
LMNA P02545 2/20 0.55
PPARG P37231 1/20 0.55
NCOA2 Q15596 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
HDAC6 Q9UBN7 1/20 0.48
TP53 P04637 1/20 0.47
CHEK1 O14757 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7050948 0.88 IKBKB (0.80) IKBKBPTPN1HPGDALDH1A1KDM4E
SCHEMBL7056469 0.88 IKBKB (0.79) IKBKBPTPN1HPGDALDH1A1KDM4E
SCHEMBL7053757 0.86 PTPN1 (0.62) IKBKBPTPN1HPGDALDH1A1KDM4E
SCHEMBL7051768 0.85 IKBKB (0.64) IKBKBPTPN1HPGDMAPT
SCHEMBL7052069 0.81 IKBKB (0.55) IKBKBPTPN1HPGDALDH1A1SMN1; SMN2
SCHEMBL7055235 0.81 CHEK1 (0.62) IKBKBPTPN1HPGDALDH1A1KDM4E
SCHEMBL7055446 0.80 IKBKB (0.72) IKBKBPTPN1HPGDALDH1A1KDM4E
SCHEMBL7057270 0.77 MAPT (0.76) IKBKBHPGDALDH1A1KDM4EMAPT
SCHEMBL23452054 0.76 KDM4E (0.61) IKBKBPTPN1HPGDALDH1A1KDM4E
SCHEMBL5361893 0.76 KDM4E (0.79) IKBKBPTPN1HPGDALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028731-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO claimed
WO-2003028731-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO disclosed