SCHEMBL7051768

SCHEMBL7051768

CNC(=O)Nc1cc(-c2ccc(N)cc2)sc1C(=O)NC

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 9/20 0.64
PTPN1 P18031 4/20 0.44
MAPK14 Q16539 3/20 0.43
RAF1 P04049 1/20 0.43
HPGD P15428 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7057485 0.85 IKBKB (0.63) IKBKBPTPN1HPGDMAPT
SCHEMBL874666 0.83 IKBKB (0.55) IKBKBPTPN1HPGDMAPT
SCHEMBL7052069 0.82 IKBKB (0.55) IKBKBPTPN1MAPK14RAF1HPGD
SCHEMBL7053757 0.80 PTPN1 (0.62) IKBKBPTPN1MAPK14RAF1HPGD
SCHEMBL7055995 0.78 CHEK1 (0.62) IKBKBMAPT
SCHEMBL7050948 0.76 IKBKB (0.80) IKBKBPTPN1HPGDMAPT
SCHEMBL7056469 0.76 IKBKB (0.79) IKBKBPTPN1HPGDMAPT
SCHEMBL7053685 0.75 IKBKB (0.78) IKBKBPTPN1HPGDMAPT
SCHEMBL7058327 0.73 IKBKB (0.58) IKBKB
SCHEMBL7057270 0.73 MAPT (0.76) IKBKBHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028731-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO disclosed