SCHEMBL7057671

SCHEMBL7057671

CNC(=O)Nc1sc(-c2ccc(N)cc2)cc1C(=O)NC.CNC(=O)Nc1sc(-c2cccc(C(F)(F)F)c2)cc1C(=O)NC

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 4/20 0.56
MAP4K4 O95819 1/20 0.56
JAK2 O60674 2/20 0.48
PIK3CD O00329 1/20 0.44
PIK3CA P42336 1/20 0.44
PIK3CG P48736 1/20 0.44
PTGS1 P23219 1/20 0.44
IKBKB O14920 1/20 0.42
CDK2AP1 O14519 1/20 0.42
KIF11 P52732 1/20 0.42
IL2 P60568 1/20 0.42
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7058130 0.94 CHEK1 (0.59) CHEK1MAP4K4JAK2PIK3CDPIK3CA
SCHEMBL7055995 0.88 CHEK1 (0.62) CHEK1MAP4K4JAK2IKBKBLMNA
SCHEMBL7052328 0.81 CHEK1 (0.78) CHEK1MAP4K4JAK2IKBKBPOLB
SCHEMBL7058543 0.79 CHEK1 (0.50) CHEK1MAP4K4IKBKBLMNAHDAC6
SCHEMBL7055932 0.78 CHEK1 (0.59) CHEK1MAP4K4JAK2IKBKBCDK2AP1
SCHEMBL7058327 0.78 IKBKB (0.58) CHEK1MAP4K4JAK2IKBKBHDAC6
SCHEMBL7057743 0.75 IKBKB (0.60) CHEK1MAP4K4JAK2IKBKBHDAC6
SCHEMBL5898639 0.74 JAK2 (0.65) CHEK1JAK2IKBKBHDAC6
SCHEMBL7051467 0.74 CHEK1 (0.56) CHEK1MAP4K4IKBKBPOLBKDM4E
SCHEMBL7053485 0.74 JAK2 (0.73) CHEK1MAP4K4JAK2IKBKBKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003029241-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO claimed