SCHEMBL7058610

SCHEMBL7058610

CS(=O)(=O)Oc1ccccc1NC1CCN(CCCCNC(=O)c2ccc(-c3cn4ccsc4n3)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 17/20 0.53
DRD2 P14416 16/20 0.53
DRD4 P21917 5/20 0.42
HTR1A P08908 3/20 0.42
HTR2A P28223 3/20 0.42
HTR2C P28335 3/20 0.42
HTR2B P41595 2/20 0.42
KCNH2 Q12809 1/20 0.41
CYP1A2 P05177 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7119545 0.92 DRD3 (0.64) DRD3DRD2DRD4HTR1AHTR2A
SCHEMBL7056847 0.87 DRD2 (0.49) DRD3DRD2DRD4HTR1AHTR2A
SCHEMBL7118079 0.81 DRD2 (0.46) DRD3DRD2DRD4HTR1AHTR2A
SCHEMBL7053088 0.78 DRD3 (0.49) DRD3DRD2DRD4HTR2ASMN1; SMN2
SCHEMBL7051851 0.78 DRD3 (0.49) DRD3DRD2DRD4HTR2ASMN1; SMN2
SCHEMBL7055489 0.76 PHF13 (0.58) DRD3DRD2DRD4CYP1A2CYP2C19
SCHEMBL7115347 0.75 DRD3 (0.49) DRD3DRD2DRD4HTR1AHTR2A
SCHEMBL7056494 0.74 DRD2 (0.60) DRD3DRD2DRD4HTR1AHTR2A
SCHEMBL7056485 0.74 DRD2 (0.64) DRD3DRD2DRD4HTR1AHTR2A
SCHEMBL7055010 0.73 DRD2 (0.61) DRD3DRD2DRD4HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028725-A1 4-(1-PIPERIDINY)-BUTYLCARBOXAMIDE AS D3 DOPAMINE RECEPTOR SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed