SCHEMBL7058824

SCHEMBL7058824

CCOC(=O)[C@@H]1C[C@@H]2CC(=O)CC[C@H]2CN1C(=O)OC

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.32
LMNA P02545 1/20 0.32
KMT2A Q03164 1/20 0.32
MAPT P10636 3/20 0.32
CYP3A4 P08684 2/20 0.32
MMP2 P08253 1/20 0.32
ANPEP P15144 1/20 0.32
TSHR P16473 2/20 0.32
FKBP1A P62942 2/20 0.32
THRB P10828 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25475425 1.00 ALDH1A1 (0.32) ALDH1A1LMNAKMT2AMAPTCYP3A4
SCHEMBL3302863 1.00 ALDH1A1 (0.32) ALDH1A1LMNAKMT2AMAPTCYP3A4
SCHEMBL8867224 0.90 MMP2 (0.39) ALDH1A1MAPTCYP3A4MMP2ANPEP
SCHEMBL8866598 0.90 MMP2 (0.39) ALDH1A1MAPTCYP3A4MMP2ANPEP
SCHEMBL3303917 0.88 MEN1 (0.36) ALDH1A1KMT2AMAPTCYP3A4TSHR
SCHEMBL24166249 0.88 MEN1 (0.36) ALDH1A1KMT2AMAPTCYP3A4TSHR
SCHEMBL6606249 0.87 ALDH1A1 (0.34) ALDH1A1LMNAKMT2AMAPTCYP3A4
SCHEMBL6611656 0.84 ALDH1A1 (0.30) ALDH1A1LMNAKMT2AMAPTCYP3A4
SCHEMBL6611658 0.84 ALDH1A1 (0.30) ALDH1A1LMNAKMT2AMAPTCYP3A4
SCHEMBL13390232 0.84 TSHR (0.36) MMP2ANPEPTSHRTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1208087-B1 DIESTER PRODRUGS OF A DECAHYDROISOQUINOLINE-3-CARBOXYLIC ACID LILLY CO ELI (US) 2003-05-14 EP disclosed
US-6486175-B1 Diester prodrugs of a decahydroisoquinoline-3-carboxylic acid ELI LILLY AND COMPANY 2002-11-26 US disclosed
US-6242462-B1 NOVEL DECAHYDROISOQUINOLINE DERIVATIVES WHICH ARE SELECTIVE GLUR5 RECEPTOR ANTAGONISTS. ELI LILLY AND COMPANY 2001-06-05 US disclosed