SCHEMBL3302863

SCHEMBL3302863

CCOC(=O)C1CC2CC(=O)CCC2CN1C(=O)OC

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.32
LMNA P02545 1/20 0.32
KMT2A Q03164 1/20 0.32
MAPT P10636 3/20 0.32
CYP3A4 P08684 2/20 0.32
MMP2 P08253 1/20 0.32
ANPEP P15144 1/20 0.32
TSHR P16473 2/20 0.32
FKBP1A P62942 2/20 0.32
THRB P10828 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7058824 1.00 ALDH1A1 (0.32) ALDH1A1LMNAKMT2AMAPTCYP3A4
SCHEMBL25475425 1.00 ALDH1A1 (0.32) ALDH1A1LMNAKMT2AMAPTCYP3A4
SCHEMBL8867224 0.90 MMP2 (0.39) ALDH1A1MAPTCYP3A4MMP2ANPEP
SCHEMBL8866598 0.90 MMP2 (0.39) ALDH1A1MAPTCYP3A4MMP2ANPEP
SCHEMBL3303917 0.88 MEN1 (0.36) ALDH1A1KMT2AMAPTCYP3A4TSHR
SCHEMBL24166249 0.88 MEN1 (0.36) ALDH1A1KMT2AMAPTCYP3A4TSHR
SCHEMBL6606249 0.87 ALDH1A1 (0.34) ALDH1A1LMNAKMT2AMAPTCYP3A4
SCHEMBL6611656 0.84 ALDH1A1 (0.30) ALDH1A1LMNAKMT2AMAPTCYP3A4
SCHEMBL6611658 0.84 ALDH1A1 (0.30) ALDH1A1LMNAKMT2AMAPTCYP3A4
SCHEMBL13390232 0.84 TSHR (0.36) MMP2ANPEPTSHRTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 52 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6939511-B2 Contact lens treating method and composition NOVARTIS AG (CH) 2005-09-06 US claimed
US-20040071591-A1 Contact lens treating method and composition ALCON INC. (CH) 2004-04-15 US claimed
US-6569824-B2 Disinfecting with an aqueous solution containing an effective amount of a monoperphthalic acid compound in a given concentration NOVARTIS AG (CH) 2003-05-27 US claimed
US-20030078171-A1 Contact lens treating method and composition ALCON INC. (CH) 2003-04-24 US claimed
EP-1255573-A1 CONTACT LENS TREATING METHOD AND COMPOSITION Novartis AG (CH) 2002-11-13 EP claimed
WO-2001060421-A1 CONTACT LENS TREATING METHOD AND COMPOSITION NOVARTIS AG (CH) 2001-08-23 WO claimed
US-20250074887-A1 PHARMACEUTICAL COMPOSITIONS OF 6-(2-(2H-TETRAZOL-5-YL)ETHYL)DECAHYDROISOQUINOLINE-3-CARBOXYLIC ACID AND DERIVATIVES THEREOF Sea Pharmaceuticals LLC. (US) 2025-03-06 US disclosed
US-20100094014-A1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS MARTINEZ-PEREZ JOSE ANTONIO 2010-04-15 US disclosed
EP-2166003-A1 Excitatory amino acid receptor antagonists Eli Lilly & Company (US) 2010-03-24 EP disclosed
US-7601738-B2 Excitatory amino acid receptor antagonists ELI LILLY AND COMPANY (US) 2009-10-13 US disclosed
EP-1368032-B1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-06-11 EP disclosed
US-7205313-B2 Excitatory amino acid receptor antagonists ELI LILLY AND COMPANY (US) 2007-04-17 US disclosed
US-20060100237-A1 Excitatory amino acid receptor antagonists ARNOLD MACKLIN B 2006-05-11 US disclosed
US-5356902-A Central nervous system disorders ELI LILLY AND COMPANY (US) 1994-10-18 US disclosed
EP-0599518-A1 Process and intermediates for the preparation of excitatory amino acide receptor antagonists ELI LILLY AND COMPANY (US) 1994-06-01 EP disclosed
EP-0590789-A1 Excitatory amino acid receptor antagonists ELI LILLY AND COMPANY (US) 1994-04-06 EP disclosed
US-5284957-A Substituted 1H- or 2H-tetrazoles ELI LILLY AND COMPANY (US) 1994-02-08 US disclosed
EP-0383504-A2 Decahydro isoquinoline derivatives, process for their preparation and use as medicines ELI LILLY AND COMPANY (US) 1990-08-22 EP disclosed
CN-1044816-A Improvements relating to organic compounds LILLY CO ELI (US) 1990-08-22 CN disclosed
US-4902695-A ISOQUINOLINE DERIVATIVES; NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1990-02-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250074887-A1 PHARMACEUTICAL COMPOSITIONS OF 6-(2-(2H-TETRAZOL-5-YL)ETHYL)DECAHYDROISOQUINOLINE-3-CARBOXYLIC ACID AND DERIVATIVES THEREOF GABRQ, GRIK5, CYP3A7 ALDH1A1 501/4885LMNA 1938/4885KMT2A 1192/4885
US-20100094014-A1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS SLC1A2, SLC1A1, GRIN1 ALDH1A1 1633/4885LMNA 2973/4885KMT2A 1887/4885
US-20060100237-A1 Excitatory amino acid receptor antagonists SLC1A2, SLC1A1, GRIN1 ALDH1A1 1633/4885LMNA 2973/4885KMT2A 1887/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.