SCHEMBL7061173

SCHEMBL7061173

COc1ccc(SCCC2CCCN2C)cc1F

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 5/20 0.46
CHRNA3 P32297 5/20 0.46
ACKR3 P25106 4/20 0.41
UHRF1 Q96T88 1/20 0.41
EHMT2 Q96KQ7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7061352 0.85 CHRM3 (0.48) ACKR3
SCHEMBL7062275 0.77 SIGMAR1 (0.44)
SCHEMBL12314795 0.75 CHRNB4 (0.45) CHRNB4CHRNA3
SCHEMBL194099 0.75 CHRNB4 (0.45) CHRNB4CHRNA3
SCHEMBL7061296 0.74 HTR6 (0.49) CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL6333252 0.74 ESRRG (0.44) CHRNB4CHRNA3
SCHEMBL7161658 0.72 CHRNB2 (0.45) CHRNB4CHRNA3
SCHEMBL11458219 0.72 CHRNB4 (0.56) CHRNB4CHRNA3EHMT2
SCHEMBL19461951 0.70 CHRNB4 (0.57) CHRNB4CHRNA3EHMT2
SCHEMBL11458400 0.70 CHRNB4 (0.54) CHRNB4CHRNA3EHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874818-B1 NOVEL SUBSTITUTED ARYL COMPOUNDS USEFUL AS MODULATORS OF ACETYLCHOLINE RECEPTORS MERCK & CO INC (US) 2003-05-21 EP disclosed
US-6316490-B1 FOR THERAPY OF PARKINSON'S DISEASE, ALZHEIMER'S DISEASE, DEMENTIA, CONTROLLING PAIN MERCK & CO., INC. 2001-11-13 US disclosed