SCHEMBL7064372

SCHEMBL7064372

CCCCCNC(=O)N(CCc1ccc(N)c(I)c1)C(=O)C(Cc1ccccc1)NC(=O)CCC(=O)OC

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 5/20 0.41
CHRNB2 P17787 2/20 0.41
CHRNB4 P30926 2/20 0.41
CHRNA3 P32297 2/20 0.41
CHRNA4 P43681 2/20 0.41
GRIA1 P42261 2/20 0.37
HPGD P15428 1/20 0.37
FAAH O00519 2/20 0.37
CHRND Q07001 5/20 0.36
CHRNA1 P02708 1/20 0.36
CHRNG P07510 1/20 0.36
CHRNB1 P11230 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7571008 0.83 PTPN1 (0.58) PTPN1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL7127958 0.76 PTPN1 (0.60) PTPN1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL29283680 0.74 CHRNB2 (0.62) PTPN1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL6831292 0.69 PTPRB (0.50) PTPN1
SCHEMBL7569835 0.68 PTPN1 (0.67) PTPN1
SCHEMBL7571014 0.68 PTPN1 (0.52) PTPN1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL7127951 0.68 CHRNB2 (0.47) PTPN1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL14113280 0.66 ACE (0.62) FAAH
SCHEMBL10655849 0.66 ACE (0.62) FAAH
SCHEMBL6918308 0.66 PTPN1 (0.69) PTPN1CHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313696-A2 AMINO(OXO)ACETIC ACID PROTEIN TYROSINE PHOSPHATASE INHIBITORS ABBOTT LABORATORIES (US) 2003-05-28 EP disclosed
WO-2002018323-A2 AMINO(OXO)ACETIC ACID PROTEIN TYROSINE PHOSPHATASE INHIBITORS ABBOTT LABORATORIES (US) 2002-03-07 WO disclosed