SCHEMBL7065623

SCHEMBL7065623

COC(=O)N(C(=O)[C@H](C)N)c1cccc2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 5/20 0.40
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
SIGMAR1 Q99720 3/20 0.40
CARM1 Q86X55 1/20 0.39
PRMT6 Q96LA8 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
RCE1 Q9Y256 1/20 0.39
GAA P10253 3/20 0.39
ALOX5 P09917 1/20 0.36
XIAP P98170 1/20 0.36
PGR P06401 1/20 0.36
PTGS1 P23219 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27532540 0.82 GAA (0.44) NCEH1ALDH1A1KDM4ESIGMAR1MEN1
SCHEMBL2090835 0.77 SIGMAR1 (0.61) NCEH1ALDH1A1SIGMAR1GAAPGR
SCHEMBL7065619 0.75 NCEH1 (0.40) NCEH1ALDH1A1KDM4ETDP1SIGMAR1
SCHEMBL7065626 0.75 NCEH1 (0.40) NCEH1ALDH1A1KDM4ETDP1SIGMAR1
SCHEMBL4847152 0.73 SMPD2 (0.44) SIGMAR1ALOX5
SCHEMBL9540683 0.73 NCEH1 (0.39) NCEH1ALDH1A1KDM4ESIGMAR1MEN1
Hydrochloric Acid SCHEMBL7437007 0.72 SMPD2 (0.43) SIGMAR1CARM1PRMT6ALOX5
SCHEMBL5558314 0.70 SIGMAR1 (0.38) ALDH1A1KDM4ESIGMAR1GAAALOX5
SCHEMBL6685262 0.70 SIGMAR1 (0.48) ALDH1A1KDM4ESIGMAR1GAAALOX5
SCHEMBL11024265 0.70 GAA (0.77) ALDH1A1KDM4ETDP1SIGMAR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313696-A2 AMINO(OXO)ACETIC ACID PROTEIN TYROSINE PHOSPHATASE INHIBITORS ABBOTT LABORATORIES (US) 2003-05-28 EP disclosed
WO-2002018323-A2 AMINO(OXO)ACETIC ACID PROTEIN TYROSINE PHOSPHATASE INHIBITORS ABBOTT LABORATORIES (US) 2002-03-07 WO disclosed