SCHEMBL7066909

SCHEMBL7066909

COC(=O)c1ccc(CNc2nc(NCc3cccs3)nc3ccsc23)cc1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.48
ADORA1 P30542 1/20 0.48
PDE4A P27815 7/20 0.46
PDE4B Q07343 7/20 0.46
PDE4C Q08493 7/20 0.46
PDE4D Q08499 7/20 0.46
ADORA2B P29275 5/20 0.46
PDE3B Q13370 4/20 0.45
PDE3A Q14432 4/20 0.45
LRRK2 Q5S007 1/20 0.44
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7071101 0.89 ADORA2A (0.53) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL7254519 0.82 NPC1 (0.52) HPGD
SCHEMBL7071277 0.82 PDE4A (0.56) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL7070989 0.81 PDE4A (0.48) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL7071479 0.81 USP1 (0.49) HPGD
SCHEMBL7071282 0.76 PDE4A (0.53) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL7254511 0.75 LMNA (0.56) HPGD
SCHEMBL7070110 0.75 LRRK2 (0.56) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL7070303 0.73 PDE4A (0.59) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL7254877 0.72 MAPT (0.50) HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003055890-A1 THIENOPYRIMIDINE DERIVATIVE COMPOUNDS AS INHIBITORS OF PROLYLPEPTIDASE, INDUCERS OF APOPTOSIS AND CANCER TREATMENT AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-10 WO disclosed