SCHEMBL7071479

SCHEMBL7071479

COC(=O)c1ccc(CNc2nc(NCc3cccs3)ncc2C)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP1 O94782 2/20 0.49
WDR48 Q8TAF3 2/20 0.49
HDAC6 Q9UBN7 2/20 0.47
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.47
ABL1 P00519 1/20 0.46
SRC P12931 1/20 0.46
HPGD P15428 2/20 0.44
POLB P06746 1/20 0.44
CLK1 P49759 1/20 0.43
CLK2 P49760 1/20 0.43
DYRK1A Q13627 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
DYRK1B Q9Y463 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
KDM4E B2RXH2 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7071470 0.90 USP1 (0.51) USP1WDR48HDAC6HDAC3HDAC1
SCHEMBL7066909 0.81 ADORA2A (0.48) HPGD
SCHEMBL7254519 0.77 NPC1 (0.52) HPGDCLK4CYP1A2CYP3A4CYP2D6
SCHEMBL7068349 0.77 CA1 (0.48) USP1WDR48ALDH1A1CA1CA2
SCHEMBL8346496 0.73 POLB (0.46) POLBALDH1A1TSHRRAB9A
SCHEMBL7257480 0.71 USP1 (0.59) USP1WDR48HPGDCLK4CYP1A2
SCHEMBL7254511 0.70 LMNA (0.56) HPGDCLK4CYP1A2CYP3A4CYP2D6
SCHEMBL1064735 0.69 CA1 (0.60) HDAC1HPGDPKMALDH1A1CA1
SCHEMBL7071101 0.69 ADORA2A (0.53)
SCHEMBL8924338 0.68 CYP4A11 (0.59) HPGDPOLBALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003055489-A1 2,4-DIAMINO-PYRIMIDINE DERIVATIVE COMPOUNDS AS INHIBITORS OF PROLYLPEPTIDASE, INDUCERS OF APOPTOSIS AND CANCER TREATMENT AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-10 WO disclosed