SCHEMBL7067258

SCHEMBL7067258

CCc1c(Sc2ccccc2)n(CC2CC=CC2)c(=O)[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
BRD4 O60885 3/20 0.35
BRDT Q58F21 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
MAPK1 P28482 3/20 0.33
PKM P14618 3/20 0.33
TSHR P16473 2/20 0.33
LMNA P02545 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.31
DHFR P00374 2/20 0.31
TYMS P04818 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7073497 0.85 GRIN1 (0.35) ALDH1A1SMN1; SMN2PKMMEN1KMT2A
SCHEMBL2470154 0.84 HPGD (0.35) ALDH1A1BRD4BRDTSMN1; SMN2MAPK1
SCHEMBL7066669 0.79 BRD4 (0.34) ALDH1A1BRD4BRDTSMN1; SMN2MAPK1
SCHEMBL7213295 0.78 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2MAPK1PKMTSHR
SCHEMBL7756601 0.77 ALDH1A1 (0.37) ALDH1A1BRD4BRDTSMN1; SMN2MAPK1
SCHEMBL7757667 0.77 LMNA (0.52) ALDH1A1SMN1; SMN2PKMTSHRLMNA
SCHEMBL599846 0.77 ALDH1A1 (0.41) ALDH1A1BRD4BRDTSMN1; SMN2MAPK1
SCHEMBL7071341 0.77 MEN1 (0.33) ALDH1A1BRD4BRDTMAPK1TSHR
SCHEMBL7756577 0.76 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2MAPK1PKMTSHR
SCHEMBL7756583 0.76 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2MAPK1PKMTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0827498-B1 NEW ANTIVIRAL SUBSTITUTED PYRIMIDINEDIONE HOMOCARBOCYCLIC NUCLEOSIDE DERIVATIVES AND METHODS FOR THE PREPARATION THEREOF AND COMPOSITIONS CONTAINING THE SAME AS ACTIVE INGREDIENTS SAMJIN PHARM CO LTD (KR) 2003-06-18 EP disclosed
US-5922727-A 1-((SUBSTITUTED)CYCLOALK(EN)YLALKYL)-6-((SUB)PHENYL(CARBONYL, SULFIDE, OR OXO))-2,4-PYRIMIDINEDIONE DERIVATIVES HAVING SUPERIOR ANTIVIRAL ACTIVITIES; HIV SAMJIN PHARMACEUTICAL CO., LTD (KR) 1999-07-13 US disclosed