SCHEMBL2470154

SCHEMBL2470154

CC(C)c1c(Sc2ccccc2)n(CC2CC=CC2)c(=O)[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.35
POLB P06746 1/20 0.35
DAO P14920 2/20 0.34
ALDH1A1 P00352 4/20 0.33
TSHR P16473 3/20 0.33
LMNA P02545 2/20 0.33
PKM P14618 1/20 0.33
MAPK1 P28482 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CXCL8 P10145 1/20 0.32
NOD2 Q9HC29 1/20 0.32
NOD1 Q9Y239 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PTPN1 P18031 1/20 0.31
CDC25A P30304 1/20 0.31
CDC25B P30305 1/20 0.31
BRD4 O60885 1/20 0.31
BRDT Q58F21 1/20 0.31
DHFR P00374 1/20 0.31
MDM2 Q00987 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7070555 0.85 GRIN1 (0.35) ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL7067258 0.84 ALDH1A1 (0.35) POLBALDH1A1TSHRLMNAPKM
SCHEMBL7070306 0.77 POLB (0.33) HPGDPOLBCXCL8NOD2NOD1
SCHEMBL2471003 0.77 GRIN1 (0.42) ALDH1A1TSHRHSD17B10MEN1KMT2A
SCHEMBL2471363 0.75 GRIN1 (0.39) POLBALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL8760732 0.75 UPP1 (0.46) HPGDPOLBALDH1A1TSHRMAPK1
SCHEMBL2471911 0.75 GRIN1 (0.39) POLBALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL7068424 0.75 TDP1 (0.33) HPGDPOLBCXCL8NOD2NOD1
SCHEMBL2469750 0.74 GRIN1 (0.38) POLBALDH1A1TSHRHSD17B10MEN1
SCHEMBL7072203 0.74 PKM (0.30) PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1986651-B1 USE OF A PYRIMIDINEDIONE DERIVATIVE FOR PREVENTING OR TREATING HEPATITIS C SAMJIN PHARM CO LTD (KR) 2011-10-05 EP claimed
US-7851479-B2 Use of pyrimidinedione derivative for preventing or treating hepatitis C SAMJIN PHARM. CO., LTD. (KR) 2010-12-14 US claimed
US-20090023764-A1 Use of Pyrimidinedione Derivative for Preventing or Treating Hepatitis C SAMJIN PHARM. CO., LTD. (KR) 2009-01-22 US claimed
US-7851479-B2 Use of pyrimidinedione derivative for preventing or treating hepatitis C SAMJIN PHARM. CO., LTD. (KR) 2010-12-14 US disclosed
US-7851479-B2 Use of pyrimidinedione derivative for preventing or treating hepatitis C SAMJIN PHARM. CO., LTD. (KR) 2010-12-14 US disclosed
US-20090023764-A1 Use of Pyrimidinedione Derivative for Preventing or Treating Hepatitis C SAMJIN PHARM. CO., LTD. (KR) 2009-01-22 US disclosed
US-20090023764-A1 Use of Pyrimidinedione Derivative for Preventing or Treating Hepatitis C SAMJIN PHARM. CO., LTD. (KR) 2009-01-22 US disclosed
US-5922727-A 1-((SUBSTITUTED)CYCLOALK(EN)YLALKYL)-6-((SUB)PHENYL(CARBONYL, SULFIDE, OR OXO))-2,4-PYRIMIDINEDIONE DERIVATIVES HAVING SUPERIOR ANTIVIRAL ACTIVITIES; HIV SAMJIN PHARMACEUTICAL CO., LTD (KR) 1999-07-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090023764-A1 Use of Pyrimidinedione Derivative for Preventing or Treating Hepatitis C DPYD, UMPS, TYMP HPGD 161/4885POLB 264/4885DAO 1357/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.