SCHEMBL7067952

SCHEMBL7067952

CC(C)(C)OC(=O)[C@]1(C)C[C@@H](C(C)(C)C)N(C(O[SiH3])(c2ccccc2)c2ccccc2)C1=O

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 1/20 0.33
LMNA P02545 1/20 0.31
CPB2 Q96IY4 2/20 0.31
GPR119 Q8TDV5 1/20 0.31
RORC P51449 7/20 0.30
KDM1A O60341 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7067547 0.73 KDM1A (0.34) GPR119RORCKDM1A
SCHEMBL7518553 0.70 GPR119 (0.34) USP30GPR119RORCKDM1A
SCHEMBL17040614 0.65 KMT2A (0.42)
SCHEMBL7067385 0.63 GPR119 (0.36) GPR119RORC
SCHEMBL7515485 0.63 GPR119 (0.36) GPR119RORC
SCHEMBL7067183 0.61 KLK7 (0.36) USP30GPR119RORCKDM1A
SCHEMBL27789215 0.60 GRIN2B (0.34) USP30
SCHEMBL13021388 0.60 KMT2A (0.41) RORC
SCHEMBL28743765 0.60 NOTUM (0.46) RORCKDM1A
SCHEMBL10920030 0.59 KCNN4 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1314041-A2 SCREEN FOR GLUTAMATE REUPTAKE INHIBITORS, STIMULATORS, AND MODULATORS Annovis, Inc. (US) 2003-05-28 EP disclosed
WO-2002018941-A2 SCREEN FOR GLUTAMATE REUPTAKE INHIBITORS, STIMULATORS, AND MODULATORS ANNOVIS, INC. (US) 2002-03-07 WO disclosed
EP-0809624-A1 ALKYLCARBOXY AMINO ACIDS-MODULATORS OF THE KAINATE RECEPTOR Bearsden Bio, Inc. (US) 1997-12-03 EP disclosed
WO-1996025387-A1 ALKYLCARBOXY AMINO ACIDS-MODULATORS OF THE KAINATE RECEPTOR SYMPHONY PHARMACEUTICALS, INC. (US) 1996-08-22 WO disclosed