SCHEMBL7069987

SCHEMBL7069987

Cc1nc(-c2ccc(N3CCNCC3)cc2)no1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52
ADRB1 P08588 5/20 0.51
DGAT1 O75907 3/20 0.50
THRB P10828 1/20 0.47
CETP P11597 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
PLK1 P53350 1/20 0.44
ACVR1 Q04771 2/20 0.44
HTR3E A5X5Y0 3/20 0.44
HTR3B O95264 3/20 0.44
HTR3A P46098 3/20 0.44
HTR3D Q70Z44 3/20 0.44
HTR3C Q8WXA8 3/20 0.44
SIGMAR1 Q99720 3/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4419949 0.99 MAOA (0.51) MAOAMAOBADRB1DGAT1THRB
SCHEMBL3074024 0.89 DGAT1 (0.58) MAOAMAOBDGAT1THRBCA12
SCHEMBL8221014 0.83 L3MBTL1 (0.59) ADRB1THRBL3MBTL1HTR3EHTR3B
SCHEMBL20076229 0.83 NR1I2 (0.44) MAOAMAOBDGAT1THRBCA12
SCHEMBL7070577 0.79 SMN1; SMN2 (0.52) MAOAMAOBSIGMAR1MAPT
SCHEMBL21956060 0.79 CETP (0.60) ADRB1CETPACVR1HTR3EHTR3B
SCHEMBL8226429 0.79 L3MBTL1 (0.46) MAOAMAOBL3MBTL1TP53MAPT
SCHEMBL8226248 0.79 L3MBTL1 (0.46) MAOAMAOBTHRBL3MBTL1MAPT
Hydrochloric Acid SCHEMBL21876097 0.77 CETP (0.59) ADRB1CETPACVR1HTR3EHTR3B
SCHEMBL13415301 0.77 L3MBTL1 (0.69) MAOAMAOBCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed
CN-1272107-A Benzamidine derivatives as factor Xa inhibitors MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed