SCHEMBL7070577

SCHEMBL7070577

Cc1nc(-c2ccc(CN3CCNCC3)cc2)no1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.52
LMNA P02545 2/20 0.52
ALDH1A1 P00352 1/20 0.52
MAPT P10636 1/20 0.52
TSHR P16473 1/20 0.52
HSD17B10 Q99714 1/20 0.52
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
KCNH2 Q12809 2/20 0.48
CYP2D6 P10635 1/20 0.48
CXCR4 P61073 8/20 0.48
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
MEN1 O00255 1/20 0.47
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
ADRA2C P18825 1/20 0.47
CCR2 P41597 1/20 0.47
CXCL12 P48061 1/20 0.47
BLM P54132 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28957460 0.86 SMN1; SMN2 (0.63) SMN1; SMN2LMNAALDH1A1MAPTTSHR
SCHEMBL5225958 0.86 SMN1; SMN2 (0.59) SMN1; SMN2LMNAALDH1A1MAPTTSHR
SCHEMBL5225149 0.85 SMN1; SMN2 (0.61) SMN1; SMN2LMNAALDH1A1MAPTTSHR
SCHEMBL5224880 0.84 SMN1; SMN2 (0.62) SMN1; SMN2LMNAALDH1A1MAPTTSHR
SCHEMBL5223197 0.82 SMN1; SMN2 (0.53) SMN1; SMN2LMNAALDH1A1MAPTTSHR
SCHEMBL7986878 0.81 MAOA (0.44) SMN1; SMN2LMNAALDH1A1MAPTTSHR
SCHEMBL7074835 0.80 KMT2A (0.58) SMN1; SMN2LMNAALDH1A1MAPTTSHR
SCHEMBL7074013 0.80 HDAC4 (0.56) LMNAMAPTTSHRMAOAMAOB
SCHEMBL7069987 0.79 MAOA (0.52) MAPTMAOAMAOBSIGMAR1
SCHEMBL7245509 0.79 CXCR1 (0.58) SMN1; SMN2ALDH1A1MAPTKCNH2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed