SCHEMBL7070294

SCHEMBL7070294

CS(=O)(=O)N1CCN(C(=O)c2ccc(C(=N)N)cc2)CC1

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.56
F10 P00742 1/20 0.56
SETD7 Q8WTS6 1/20 0.55
MAPK1 P28482 1/20 0.55
ALDH1A1 P00352 2/20 0.54
HTT P42858 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
TSHR P16473 2/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
TP53 P04637 1/20 0.50
EPHX2 P34913 1/20 0.49
LMNA P02545 1/20 0.49
F11 P03951 1/20 0.48
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL27568113 0.96 GAA (0.56) GAAF10SETD7MAPK1ALDH1A1
SCHEMBL4003521 0.84 CA12 (0.65) GAASETD7MAPK1ALDH1A1HTT
SCHEMBL7069792 0.84 F10 (0.53) GAAF10ALDH1A1SMN1; SMN2TSHR
SCHEMBL12302056 0.83 MEN1 (0.70) GAASETD7MAPK1ALDH1A1HTT
SCHEMBL24064947 0.82 F11 (0.55) ALDH1A1MEN1KMT2AF11
SCHEMBL7074218 0.82 ALDH1A1 (0.67) GAAMAPK1ALDH1A1HTTSMN1; SMN2
SCHEMBL7074838 0.82 F10 (0.54) GAAF10ALDH1A1SMN1; SMN2TSHR
SCHEMBL13268583 0.81 CA12 (0.63) GAASETD7MAPK1ALDH1A1HTT
SCHEMBL2474167 0.81 GAA (0.59) GAASETD7MAPK1ALDH1A1HTT
SCHEMBL7076666 0.81 LMNA (0.72) GAAF10MAPK1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed