SCHEMBL7070692

SCHEMBL7070692

CCn1c(=O)n(C2CCN(Cc3cccc(Oc4ccccc4OC)c3)CC2)c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.57
CYP3A4 P08684 2/20 0.56
CYP2D6 P10635 2/20 0.56
CCR8 P51685 8/20 0.55
OPRL1 P41146 3/20 0.51
OPRK1 P41145 1/20 0.51
DRD2 P14416 1/20 0.50
DRD4 P21917 1/20 0.50
C5AR1 P21730 3/20 0.49
KCNH2 Q12809 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7066463 0.93 CYP3A4 (0.62) OPRM1CYP3A4CYP2D6CCR8OPRL1
SCHEMBL6496325 0.89 KDM4E (0.58) OPRM1CYP3A4CYP2D6CCR8OPRL1
SCHEMBL7068005 0.82 OPRM1 (0.84) OPRM1CCR8OPRL1OPRK1DRD2
SCHEMBL6499178 0.80 CACNA1G (0.61) OPRM1CYP3A4CYP2D6CCR8OPRL1
SCHEMBL6499157 0.79 OPRM1 (0.64) OPRM1CCR8OPRL1OPRK1DRD2
SCHEMBL6501702 0.79 CYP3A4 (0.56) OPRM1CYP3A4CYP2D6CCR8OPRL1
SCHEMBL6504157 0.79 CCR8 (0.66) CCR8KCNH2
SCHEMBL7066869 0.78 OPRM1 (0.51) OPRM1CYP3A4CYP2D6CCR8OPRL1
SCHEMBL6505921 0.77 C5AR1 (0.57) OPRM1CYP3A4CYP2D6CCR8OPRL1
SCHEMBL6495959 0.77 CYP3A4 (0.53) OPRM1CYP3A4CYP2D6CCR8OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003037271-A2 COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE THEREFOR MILLENNIUM PHARMACEUTICALS,INC. (US) 2003-05-08 WO disclosed