SCHEMBL7071995

SCHEMBL7071995

Cn1cccc1-c1nc2c[nH]c(N)nc-2n1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.37
NPC1 O15118 2/20 0.37
RECQL P46063 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ALDH1A1 P00352 4/20 0.35
GAA P10253 1/20 0.35
ALOX15 P16050 1/20 0.35
CYP2A6 P11509 1/20 0.34
CYP2A13 Q16696 1/20 0.34
HSD17B10 Q99714 2/20 0.33
MAPK1 P28482 2/20 0.33
PCSK9 Q8NBP7 1/20 0.32
MEN1 O00255 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30
MAPT P10636 2/20 0.30
LMNA P02545 1/20 0.30
TSHR P16473 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7077154 0.78 HTR6 (0.41) PCSK9
SCHEMBL18482878 0.71 ALDH1A1 (0.47) KDM4ENPC1RECQLNPSR1ALDH1A1
SCHEMBL2115936 0.68 ALDH1A1 (0.41) KDM4ENPC1RECQLNPSR1ALDH1A1
SCHEMBL18483370 0.67 ALDH1A1 (0.40) KDM4ENPC1RECQLNPSR1ALDH1A1
SCHEMBL18471452 0.67 ALDH1A1 (0.40) KDM4ENPC1RECQLNPSR1ALDH1A1
SCHEMBL3469899 0.66 KDM4E (0.42) KDM4ENPC1RECQLNPSR1ALDH1A1
SCHEMBL1232645 0.66 KDM4E (0.45) KDM4ENPC1RECQLNPSR1ALDH1A1
SCHEMBL7070801 0.66 ADORA2A (0.44) KDM4ENPC1RECQLALDH1A1ALOX15
SCHEMBL2117930 0.65 ALDH1A1 (0.41) KDM4ENPC1RECQLNPSR1ALDH1A1
SCHEMBL3268785 0.64 KDM4E (0.38) KDM4ENPC1RECQLNPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed