SCHEMBL7073236

SCHEMBL7073236

COc1ccc(CBr)c(C(=O)O)c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.54
POLB P06746 6/20 0.54
KDM4E B2RXH2 5/20 0.54
AKR1C3 P42330 5/20 0.47
AKR1C2 P52895 5/20 0.47
ALDH1A1 P00352 5/20 0.46
HSD17B10 Q99714 2/20 0.46
LMNA P02545 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
NPC1 O15118 1/20 0.46
APEX1 P27695 1/20 0.46
RAB9A P51151 1/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
HPGD P15428 2/20 0.45
SLC16A3 O15427 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2317055 0.86 AKR1C3 (0.50) SMN1; SMN2POLBKDM4EAKR1C3AKR1C2
SCHEMBL10112008 0.86 ALDH1A1 (0.54) SMN1; SMN2POLBKDM4EALDH1A1HSD17B10
SCHEMBL13469239 0.86 SMN1; SMN2 (0.57) SMN1; SMN2POLBKDM4EAKR1C3AKR1C2
SCHEMBL149036 0.85 KDM4E (0.55) SMN1; SMN2POLBKDM4EALDH1A1HSD17B10
SCHEMBL8482547 0.84 SMN1; SMN2 (0.56) SMN1; SMN2POLBKDM4EAKR1C3AKR1C2
SCHEMBL8482552 0.84 SMN1; SMN2 (0.60) SMN1; SMN2POLBKDM4EAKR1C3AKR1C2
SCHEMBL11608784 0.83 KDM4E (0.50) SMN1; SMN2KDM4EAKR1C3AKR1C2ALDH1A1
SCHEMBL8338550 0.83 SMN1; SMN2 (0.54) SMN1; SMN2POLBKDM4EAKR1C3AKR1C2
SCHEMBL1399960 0.83 HSD17B10 (0.63) SMN1; SMN2POLBKDM4EAKR1C3AKR1C2
SCHEMBL18280327 0.83 SMN1; SMN2 (0.54) SMN1; SMN2POLBKDM4EAKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3924349-B1 AMINO ACID DERIVATIVES FOR THE TREATMENT OF INFLAMMATORY DISEASES THE ROSKAMP INST (US) 2025-06-25 EP disclosed
EP-3303415-B1 VISIBLE-LIGHT PHOTOINITIATORS AND USES THEREOF ALCON INC (CH) 2022-12-28 EP disclosed
US-20220081415-A1 Amino Acid Derivatives for the Treatment of Inflammatory Diseases THE ROSKAMP INST (US) 2022-03-17 US disclosed
EP-3924349-A2 AMINO ACID DERIVATIVES FOR THE TREATMENT OF INFLAMMATORY DISEASES The Roskamp Institute (US) 2021-12-22 EP disclosed
CN-113614074-A Amino acid derivatives for the treatment of inflammatory diseases 罗斯坎普研究所 2021-11-05 CN disclosed
US-10324311-B2 Visible-light photoinitiators and uses thereof NOVARTIS AG (CH) 2019-06-18 US disclosed
EP-3303415-A1 VISIBLE-LIGHT PHOTOINITIATORS AND USES THEREOF Novartis AG (CH) 2018-04-11 EP disclosed
US-20160357031-A1 VISIBLE-LIGHT PHOTOINITIATORS AND USES THEREOF ALCON INC. (CH) 2016-12-08 US disclosed
WO-2016193912-A1 VISIBLE-LIGHT PHOTOINITIATORS AND USES THEREOF NOVARTIS AG (CH) 2016-12-08 WO disclosed
EP-0832891-B1 Dihydrobenzo (B) indeno (2,1-D) thiophene compounds, intermediates, processes, compositions, and methods LILLY CO ELI (US) 2003-07-30 EP disclosed
EP-0832890-B1 Benzo (B) indeno (2,1-D) thiophene compounds, intermediates, processes, compositions, and methods LILLY CO ELI (US) 2003-07-02 EP disclosed
US-6133458-A FOR INHIBITING BONE LOSS OR BONE RESORPTION, PARTICULARLY OSTEOPOROSIS, CARDIOVASCULAR-RELATED PATHOLOGICAL CONDITIONS INCLUDING HYPERLIPIDEMIA AND RELATED CARDIOVASCULAR PATHOLOGIES, AND ESTROGEN-DEPENDENT CANCER ELI LILLY AND COMPANY (US) 2000-10-17 US disclosed
US-5856341-A INHIBITING BONE LOSS OR BONE RESORPTION, PARTICULARLY OSTEOPOROSIS, CARDIOVASCULAR-RELATED PATHOLOGICAL CONDITIONS INCLUDING HYPERLIPIDEMIA, ESTROGEN-DEPENDENT CANCER ELI LILLY AND COMPANY (US) 1999-01-05 US disclosed
US-5834488-A INHIBIT BONE LOSS OR BONE RESORPTION, LOWER SERUM CHOLESTEROL LEVELS, INHIBIT ESTROGEN-DEPENDENT CANCER ELI LILLY AND COMPANY (US) 1998-11-10 US disclosed
EP-0832890-A1 Benzo (B) indeno (2,1-D) thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-01 EP disclosed
EP-0832891-A1 Dihydrobenzo (B) indeno (2,1-D) thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10324311-B2 Visible-light photoinitiators and uses thereof SIRT5, IK, IGLV6-57 SMN1; SMN2 4875/4885POLB 2831/4885KDM4E 389/4885
US-20160357031-A1 VISIBLE-LIGHT PHOTOINITIATORS AND USES THEREOF SIRT5, IK, IGLV6-57 SMN1; SMN2 4875/4885POLB 2831/4885KDM4E 389/4885
US-20220081415-A1 Amino Acid Derivatives for the Treatment of Inflammatory Diseases NFKBIA, NFRKB, IKBKG SMN1; SMN2 3021/4885POLB 634/4885KDM4E 1742/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.