SCHEMBL7074013

SCHEMBL7074013

Cc1nc(-c2ccc(CC(=O)N3CCNCC3)cc2)no1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.56
HDAC6 Q9UBN7 2/20 0.56
DGAT1 O75907 2/20 0.54
LMNA P02545 4/20 0.48
TSHR P16473 2/20 0.48
ALOX15 P16050 1/20 0.48
MAPK1 P28482 1/20 0.48
PLK1 P53350 1/20 0.47
HPGD P15428 1/20 0.46
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45
KCNH2 Q12809 1/20 0.44
GPR119 Q8TDV5 1/20 0.44
NFKB1 P19838 1/20 0.43
RAB9A P51151 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
MAPT P10636 2/20 0.43
HTT P42858 1/20 0.43
MGLL Q99685 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7071693 0.90 LMNA (0.55) HDAC4HDAC6DGAT1LMNATSHR
SCHEMBL7074627 0.84 TSHR (0.57) HDAC4HDAC6DGAT1LMNATSHR
SCHEMBL7074241 0.82 HDAC4 (0.53) HDAC4HDAC6DGAT1LMNAALOX15
SCHEMBL7074802 0.81 HDAC4 (0.53) HDAC4HDAC6DGAT1LMNATSHR
SCHEMBL7070577 0.80 SMN1; SMN2 (0.52) LMNATSHRMAOAMAOBKCNH2
SCHEMBL7074329 0.80 MAPT (0.59) DGAT1LMNATSHRMAPK1PLK1
SCHEMBL7069975 0.80 GAA (0.60) HDAC4HDAC6DGAT1LMNATSHR
SCHEMBL7651866 0.79 DGAT1 (0.42) DGAT1LMNATSHRMAPK1PLK1
SCHEMBL7076669 0.79 GAA (0.53) HDAC4HDAC6DGAT1LMNATSHR
SCHEMBL7074862 0.79 DGAT1 (0.53) HDAC4HDAC6DGAT1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed