SCHEMBL7651866

SCHEMBL7651866

COC(=O)C(CC(=O)N1CCNCC1)c1ccc(-c2noc(C)n2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 2/20 0.42
PLK1 P53350 1/20 0.41
MAPT P10636 7/20 0.41
TP53 P04637 3/20 0.41
POLB P06746 2/20 0.41
LMNA P02545 6/20 0.39
HPGD P15428 3/20 0.39
HTT P42858 2/20 0.39
ALDH1A1 P00352 2/20 0.39
NPC1 O15118 1/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
RAB9A P51151 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
GPR119 Q8TDV5 1/20 0.38
P2RX3 P56373 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7649098 0.85 GPR119 (0.54) DGAT1MAPTTP53POLBLMNA
SCHEMBL7074013 0.79 HDAC4 (0.56) DGAT1PLK1MAPTPOLBLMNA
SCHEMBL7649437 0.78 PKM (0.46) MAPTTP53POLBLMNAALDH1A1
SCHEMBL7071693 0.76 LMNA (0.55) DGAT1PLK1MAPTPOLBLMNA
SCHEMBL7074329 0.73 MAPT (0.59) DGAT1PLK1MAPTPOLBLMNA
SCHEMBL7655612 0.69 MAOA (0.42) DGAT1PLK1MAPTLMNAHPGD
SCHEMBL7069987 0.67 MAOA (0.52) DGAT1PLK1MAPTTP53MAOA
SCHEMBL7076934 0.67 L3MBTL1 (0.54) LMNA
SCHEMBL7070577 0.67 SMN1; SMN2 (0.52) MAPTPOLBLMNAHTTALDH1A1
Hydrochloric Acid SCHEMBL4419949 0.66 MAOA (0.51) DGAT1PLK1MAPTTP53MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed