SCHEMBL7074313

SCHEMBL7074313

N=C(N)c1ccc(C(=O)N2CCN(C(=O)Cc3ccc(Cl)cc3)CC2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
FNTA P49354 1/20 0.59
FNTB P49356 1/20 0.59
F2 P00734 1/20 0.57
PRSS1 P07477 1/20 0.57
TPSAB1 Q15661 1/20 0.57
TPSD1 Q9BZJ3 1/20 0.57
TPSG1 Q9NRR2 1/20 0.57
GFER P55789 1/20 0.53
ATM Q13315 1/20 0.53
GPR183 P32249 1/20 0.52
ME2 P23368 1/20 0.52
ME1 P48163 1/20 0.52
ME3 Q16798 1/20 0.52
ITGB3 P05106 3/20 0.52
ITGA2B P08514 3/20 0.52
POLB P06746 1/20 0.51
ALDH1A1 P00352 2/20 0.51
GAA P10253 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL28743988 0.95 CYP2C9 (0.55) CYP2C9CYP2C19FNTAFNTBF2
SCHEMBL16599088 0.84 GPR183 (0.73) CYP2C9CYP2C19FNTAFNTBGFER
SCHEMBL7075152 0.78 CNR1 (0.51) CYP2C19F2PRSS1TPSAB1TPSD1
SCHEMBL7074218 0.76 ALDH1A1 (0.67) F2PRSS1TPSAB1TPSD1TPSG1
SCHEMBL10722382 0.76 POLB (0.81) GPR183POLBALDH1A1GAAKMT2A
SCHEMBL9585721 0.76 POLB (0.81) GPR183POLBALDH1A1GAAKMT2A
SCHEMBL7077553 0.75 F10 (0.65) POLBKMT2AMEN1LMNAMAPT
SCHEMBL7430480 0.75 HPGD (0.67) CYP2C9CYP2C19GFERATMGPR183
SCHEMBL7069339 0.74 CNR1 (0.55) F2PRSS1TPSAB1TPSD1TPSG1
SCHEMBL7838912 0.74 BLM (0.71) FNTAFNTBGPR183POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed