SCHEMBL7074835

SCHEMBL7074835

Cc1nc(-c2ccc(CN3CCN(Cc4ccc5ccccc5c4)CC3)cc2)no1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.58
ALDH1A1 P00352 2/20 0.57
MAPT P10636 2/20 0.57
TSHR P16473 2/20 0.57
LMNA P02545 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
HSD17B10 Q99714 1/20 0.57
CYP2D6 P10635 1/20 0.53
KCNH2 Q12809 1/20 0.53
CHKA P35790 1/20 0.51
ACHE P22303 1/20 0.50
PKM P14618 1/20 0.50
MC4R P32245 1/20 0.47
MC5R P33032 1/20 0.47
S1PR1 P21453 2/20 0.46
OPRL1 P41146 1/20 0.46
MEN1 O00255 1/20 0.45
HTT P42858 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
DRD2 P14416 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7999722 0.88 ALDH1A1 (0.45) KMT2AALDH1A1MAPTTSHRLMNA
SCHEMBL7071609 0.86 NPC1 (0.65) KMT2AALDH1A1MAPTTSHRLMNA
SCHEMBL7074071 0.85 KDM4E (0.56) KMT2AALDH1A1MAPTTSHRLMNA
SCHEMBL7996221 0.82 PLA2G2A (0.42) KMT2AALDH1A1MAPTTSHRLMNA
SCHEMBL7073968 0.82 MAPT (0.50) KMT2AALDH1A1MAPTTSHRLMNA
SCHEMBL28957460 0.82 SMN1; SMN2 (0.63) ALDH1A1MAPTTSHRLMNASMN1; SMN2
SCHEMBL5225958 0.82 SMN1; SMN2 (0.59) ALDH1A1MAPTTSHRLMNASMN1; SMN2
SCHEMBL5225149 0.81 SMN1; SMN2 (0.61) ALDH1A1MAPTTSHRLMNASMN1; SMN2
SCHEMBL5223197 0.80 SMN1; SMN2 (0.53) ALDH1A1MAPTTSHRLMNASMN1; SMN2
SCHEMBL5224880 0.80 SMN1; SMN2 (0.62) KMT2AALDH1A1MAPTTSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed