SCHEMBL7074071

SCHEMBL7074071

Cc1nc(-c2ccc(CN3CCN(S(=O)(=O)c4ccc5ccccc5c4)CC3)cc2)no1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.56
ALDH1A1 P00352 2/20 0.56
SLC2A1 P11166 1/20 0.53
GAA P10253 1/20 0.52
LMNA P02545 5/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
PKM P14618 2/20 0.51
HTT P42858 1/20 0.48
MAPT P10636 3/20 0.48
HSD11B1 P28845 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
TSHR P16473 1/20 0.47
HSD17B10 Q99714 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7076926 0.91 LSS (0.52) KDM4EALDH1A1LMNASMN1; SMN2MAPT
SCHEMBL7070554 0.90 MAPT (0.52) KDM4EALDH1A1SLC2A1LMNASMN1; SMN2
SCHEMBL7069980 0.89 TSHR (0.54) ALDH1A1LMNASMN1; SMN2MAPTTSHR
SCHEMBL7996072 0.86 LMNA (0.46) KDM4EALDH1A1GAALMNASMN1; SMN2
SCHEMBL7074835 0.85 KMT2A (0.58) ALDH1A1LMNASMN1; SMN2PKMHTT
SCHEMBL7075159 0.85 LSS (0.51) ALDH1A1LMNASMN1; SMN2PKMHTT
SCHEMBL7074079 0.85 ALDH1A1 (0.63) KDM4EALDH1A1LMNASMN1; SMN2PKM
SCHEMBL7069977 0.85 PKM (0.55) KDM4EALDH1A1GAALMNASMN1; SMN2
SCHEMBL7074028 0.85 MAPT (0.62) KDM4ELMNASMN1; SMN2PKMHTT
SCHEMBL7076863 0.84 LSS (0.49) ALDH1A1LMNASMN1; SMN2MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed