SCHEMBL7075112

SCHEMBL7075112

CN(C)c1cccc2c(S(=O)(=O)N3CCN(C(=O)c4ccc(C(=N)N)cc4)CC3)cccc12

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.59
ATM Q13315 1/20 0.59
TGM2 P21980 5/20 0.55
F10 P00742 2/20 0.51
SPR P35270 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
F2 P00734 3/20 0.45
PRSS1 P07477 3/20 0.45
PRSS2 P07478 3/20 0.45
PRSS3 P35030 3/20 0.45
CA2 P00918 1/20 0.44
LMNA P02545 2/20 0.43
EPHX1 P07099 1/20 0.43
EPHX2 P34913 1/20 0.43
MMP2 P08253 1/20 0.43
MMP13 P45452 1/20 0.43
HTR6 P50406 1/20 0.42
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL27530351 0.97 KMT2A (0.56) KMT2AATMTGM2F10SPR
SCHEMBL7074199 0.87 TGM2 (0.58) KMT2AATMTGM2F10SPR
SCHEMBL7071342 0.85 CNR1 (0.57) KMT2AATMTGM2F10LMNA
Acetic Acid SCHEMBL27538655 0.83 CNR1 (0.53) KMT2ATGM2F10SPRSMN1; SMN2
SCHEMBL18711519 0.81 KMT2A (0.71) KMT2AATMTGM2SPRSMN1; SMN2
SCHEMBL27571758 0.81 KMT2A (0.71) KMT2AATMTGM2SPRSMN1; SMN2
SCHEMBL25531 0.80 KMT2A (0.88) KMT2AATMTGM2SMN1; SMN2F2
SCHEMBL29437927 0.80 KMT2A (0.88) KMT2AATMTGM2SMN1; SMN2F2
SCHEMBL17076474 0.79 TGM2 (0.68) KMT2AATMTGM2F10SPR
SCHEMBL7076710 0.79 MGLL (0.51) KMT2AATMTGM2SPRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed