SCHEMBL7076142

SCHEMBL7076142

O=C(O)c1cc2ccccc2n1Cc1cc2c(cc1Cl)OCO2

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 10/20 0.60
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
POLB P06746 1/20 0.45
MCL1 Q07820 2/20 0.44
GPR35 Q9HC97 1/20 0.44
TRAP1 Q12931 1/20 0.43
SLC22A12 Q96S37 1/20 0.43
EDNRB P24530 1/20 0.43
EDNRA P25101 1/20 0.43
DAO P14920 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7489141 0.86 CCR2 (0.60) CCR2GPR35TRAP1
SCHEMBL6302551 0.85 CCR2 (0.60) CCR2TRAP1SLC22A12
SCHEMBL6306908 0.85 CCR2 (0.60) CCR2ALDH1A1
SCHEMBL7465471 0.83 SRD5A2 (0.54) CCR2EDNRBEDNRA
SCHEMBL7464523 0.82 CCR2 (0.48) CCR2GPR35
SCHEMBL8388354 0.81 CCR2 (0.48) CCR2MCL1EDNRBEDNRA
SCHEMBL7469052 0.81 CCR2 (0.48) CCR2MCL1EDNRBEDNRA
SCHEMBL3966109 0.81 CCR2 (0.78) CCR2ALDH1A1CYP1A2POLBMCL1
SCHEMBL7498811 0.81 CCR2 (0.49) CCR2ALDH1A1
SCHEMBL3963211 0.80 CCR2 (0.73) CCR2ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003504-B1 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 ANTAGONISTS ASTRAZENECA AB (SE) 2003-07-02 EP disclosed