SCHEMBL7469052

SCHEMBL7469052

C[C@@H](Oc1ccc2c(c1)cc(C(=O)O)n2Cc1cc2c(cc1Cl)OCO2)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 13/20 0.48
ABCB11 O95342 2/20 0.47
S1PR5 Q9H228 2/20 0.42
S1PR1 P21453 1/20 0.42
PLA2G4A P47712 1/20 0.40
EDNRB P24530 1/20 0.38
EDNRA P25101 1/20 0.38
MCL1 Q07820 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8388354 1.00 CCR2 (0.48) CCR2ABCB11S1PR5S1PR1PLA2G4A
SCHEMBL7470926 0.87 CCR2 (0.44) CCR2ABCB11S1PR5S1PR1PLA2G4A
SCHEMBL7473359 0.87 CCR2 (0.44) CCR2ABCB11S1PR5S1PR1PLA2G4A
SCHEMBL7465471 0.83 SRD5A2 (0.54) CCR2ABCB11S1PR5S1PR1PLA2G4A
SCHEMBL7461617 0.82 CCR2 (0.41) CCR2ABCB11PLA2G4A
SCHEMBL7076142 0.81 CCR2 (0.60) CCR2EDNRBEDNRAMCL1
SCHEMBL7466879 0.81 EDNRB (0.48) CCR2ABCB11PLA2G4AEDNRBEDNRA
SCHEMBL7472885 0.81 CCR2 (0.48) CCR2ABCB11S1PR5S1PR1PLA2G4A
SCHEMBL7455739 0.79 CCR2 (0.57) CCR2ABCB11PLA2G4AEDNRBEDNRA
SCHEMBL7489141 0.79 CCR2 (0.60) CCR2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1021181-A4 CARBOXYLIC ACID INDOLE INHIBITORS OF CHEMOKINES SMITHKLINE BEECHAM CORP (US) 2002-06-26 EP disclosed
EP-1021181-A1 CARBOXYLIC ACID INDOLE INHIBITORS OF CHEMOKINES SMITHKLINE BEECHAM CORPORATION (US) 2000-07-26 EP disclosed
WO-1997035572-A1 CARBOXYLIC ACID INDOLE INHIBITORS OF CHEMOKINES SMITHKLINE BEECHAM CORPORATION (US) 1997-10-02 WO disclosed