SCHEMBL7078795

SCHEMBL7078795

CCOC(OCC)c1ccc(CC(COCc2ccccc2)(COCc2ccccc2)Cc2ccc([S+](C)[O-])cc2)cc1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.33
ACHE P22303 2/20 0.33
FFAR1 O14842 1/20 0.32
KDM4E B2RXH2 1/20 0.32
POLB P06746 1/20 0.32
PTPRB P23467 1/20 0.31
PTGS2 P35354 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6944045 0.85 MEN1 (0.37) BCHEACHEFFAR1KDM4EPOLB
SCHEMBL6950120 0.78 PTPRB (0.34) KDM4EPOLBPTPRBTSHR
SCHEMBL7137466 0.77 ALDH1A1 (0.38) BCHEACHEFFAR1KDM4EPOLB
SCHEMBL6948228 0.69 KDM4E (0.37) KDM4EPOLBPTPRBTSHR
SCHEMBL9548555 0.69 ACHE (0.46) BCHEACHEFFAR1PTGS2TSHR
SCHEMBL4661710 0.68 L3MBTL1 (0.52) BCHEACHETSHR
SCHEMBL1791345 0.67 SLC6A2 (0.43) KDM4EPOLBTSHR
SCHEMBL866663 0.67 TSHR (0.42) TSHR
SCHEMBL6948598 0.66 ACHE (0.44) BCHEACHEFFAR1PTGS2
SCHEMBL29171867 0.66 NAAA (0.42) BCHEACHEFFAR1PTGS2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115729-B1 PHOSPHONIC ACID DERIVATIVES AS INHIBITORS OF PTP-1B MERCK FROSST CANADA INC (CA) 2003-02-19 EP disclosed
US-6174874-B1 ANTIDIABETIC,-CARCINOGENIC AGENTS; IMPROVING GLUCOSE TOLERANCE/INSULIN-SENSITIVITY; PREVENTING/TREATING OBESITY AND NEURODEGENERATIVE DISEASES; E.G. 1,3-BIS-((PHOSPHONODI-FLUOROMETHYL)PHENYL)-2-DICARBOXYPROPANE MERCK FROSST CANADA & CO. (CA) 2001-01-16 US disclosed