SCHEMBL7079357

SCHEMBL7079357

COC(=O)C1CCCC1O

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.47
CHRM4 P08173 1/20 0.47
CHRM3 P20309 1/20 0.47
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2693326 1.00 CHRM2 (0.47) CHRM2CHRM4CHRM3SLC6A2SLC6A4
SCHEMBL2693319 1.00 CHRM2 (0.47) CHRM2CHRM4CHRM3SLC6A2SLC6A4
SCHEMBL2691303 1.00 CHRM2 (0.47) CHRM2CHRM4CHRM3SLC6A2SLC6A4
SCHEMBL7191976 1.00 CHRM2 (0.47) CHRM2CHRM4CHRM3SLC6A2SLC6A4
SCHEMBL8384596 1.00 CHRM2 (0.47) CHRM2CHRM4CHRM3SLC6A2SLC6A4
SCHEMBL23921599 1.00 CHRM2 (0.47) CHRM2CHRM4CHRM3SLC6A2SLC6A4
SCHEMBL10389540 0.95 CHRM2 (0.43) CHRM2CHRM4CHRM3SLC6A2SLC6A4
SCHEMBL27265137 0.95 CHRM2 (0.43) CHRM2CHRM4CHRM3SLC6A2SLC6A4
SCHEMBL262052 0.95 CHRM2 (0.43) CHRM2CHRM4CHRM3SLC6A2SLC6A4
SCHEMBL12948024 0.95 CHRM2 (0.43) CHRM2CHRM4CHRM3SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250295798-A1 LIGAND-DRUG CONJUGATE OF EXATECAN ANALOGUE, AND MEDICAL USE THEREOF BEIGENE SWITZERLAND GMBH (CH) 2025-09-25 US disclosed
EP-4594327-A1 LIGAND-DRUG CONJUGATE OF EXATECAN ANALOGUE, AND MEDICAL USE THEREOF BeiGene Switzerland GmbH (CH) 2025-08-06 EP disclosed
CN-119948031-A Ligand-drug conjugates of isatecan analogs and medical uses thereof 广州百济神州生物制药有限公司 2025-05-06 CN disclosed
US-20240376059-A1 Compounds for the Treatment of Alzheimer's Disease THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2024-11-14 US disclosed
WO-2024067811-A1 LIGAND-DRUG CONJUGATE OF EXATECAN ANALOGUE, AND MEDICAL USE THEREOF BEIGENE, LTD. (KY) 2024-04-04 WO disclosed
US-11939302-B2 Compounds for the treatment of Alzheimer's disease THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2024-03-26 US disclosed
WO-2024057013-A1 NLRP3 MODULATORS EXSCIENTIA AI LIMITED (GB) 2024-03-21 WO disclosed
CN-117447359-A Preparation method of high-purity peramivir intermediate 浙江诚意药业股份有限公司 2024-01-26 CN disclosed
CN-117250295-A Detection method of peramivir intermediate 浙江诚意药业股份有限公司 2023-12-19 CN disclosed
US-20230302162-A1 RADIOLABELED DARAPLADIB AND ANALOGS THEREOF AND THEIR USE AS IMAGING COMPOUNDS INSERM (INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE) (FR) 2023-09-28 US disclosed
US-6077958-A Heteroaromatic diphosphines as chiral ligands ITALFARMACO SUD S.P.A. (IT) 2000-06-20 US disclosed
EP-0770085-B1 HETEROAROMATIC DIPHOSPHINES AS CHIRAL LIGANDS CHEMI SPA (IT) 1999-09-22 EP disclosed
US-5907045-A Heteroaromatic diphosphines as chiral ligands ITALFARMACO SUD S.P.A. (IT) 1999-05-25 US disclosed
EP-0738254-B1 ASYMETRIC HYDROGENATION OF BETA- or GAMMA-KETOESTERS AND BETA- or GAMMA-KETOAMIDES MERCK & CO INC (US) 1999-04-14 EP disclosed
EP-0770085-A1 HETEROAROMATIC DIPHOSPHINES AS CHIRAL LIGANDS ITALFARMACO SUD S.p.A. (IT) 1997-05-02 EP disclosed
US-5596113-A HYDROGENATION CATALYSTS MERCK & CO., INC. (US) 1997-01-21 US disclosed
US-5508435-A ASYMMETRIC REDUCTION WITH A RUTHENIUM CATALYST IN PRESENCE OF A STRONG ACID MERCK & CO., INC. (US) 1996-04-16 US disclosed
WO-1996001831-A1 HETEROAROMATIC DIPHOSPHINES AS CHIRAL LIGANDS ITALFARMACO SUD S.P.A. (IT) 1996-01-25 WO disclosed
WO-1995018784-A1 ASYMETRIC HYDROGENATION OF β- or ηg-KETOESTERS AND β- or η-KETOAMIDES MERCK & CO., INC. (US) 1995-07-13 WO disclosed
US-4973354-A AGRICULTURE, OPTICAL ISOMERS NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1990-11-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250295798-A1 LIGAND-DRUG CONJUGATE OF EXATECAN ANALOGUE, AND MEDICAL USE THEREOF SLC10A1, ERBB3, SLC10A2 CHRM2 1846/4885CHRM4 1826/4885CHRM3 1142/4885
US-20240376059-A1 Compounds for the Treatment of Alzheimer's Disease IAPP, GPR119, APP CHRM2 77/4885CHRM4 76/4885CHRM3 47/4885
US-11939302-B2 Compounds for the treatment of Alzheimer's disease IAPP, GPR119, APP CHRM2 77/4885CHRM4 76/4885CHRM3 47/4885
US-20230302162-A1 RADIOLABELED DARAPLADIB AND ANALOGS THEREOF AND THEIR USE AS IMAGING COMPOUNDS PLA2G4B, PLA2G1B, PLA2G12B CHRM2 3365/4885CHRM4 4050/4885CHRM3 3856/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.