SCHEMBL7079754

SCHEMBL7079754

CC(=O)OC(Cc1cccnc1)c1nc(C(C)C)c(Sc2cc(F)cc(F)c2)[nH]1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 6/20 0.37
GRM2 Q14416 2/20 0.34
RORC P51449 1/20 0.34
NAMPT P43490 3/20 0.33
KDM4E B2RXH2 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TBXAS1 P24557 2/20 0.32
KMT2A Q03164 1/20 0.32
CYP3A4 P08684 1/20 0.32
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972343 0.93 IDO1 (0.36) IDO1GRM2RORCNAMPTKDM4E
SCHEMBL7082209 0.90 IDO1 (0.34) IDO1GRM2RORCNAMPTKDM4E
SCHEMBL6973278 0.89 MEN1 (0.35) IDO1RORCNAMPTKDM4EHSD17B10
SCHEMBL6969311 0.89 LMNA (0.37) IDO1NAMPTKDM4EHSD17B10TBXAS1
SCHEMBL6973902 0.87 IDO1 (0.32) IDO1GRM2RORC
SCHEMBL6967430 0.86 ALDH1A1 (0.41) IDO1RORCKDM4EKMT2A
SCHEMBL6969546 0.86 IDO1 (0.36) IDO1GRM2RORCNAMPTKDM4E
SCHEMBL6973462 0.84 ALDH1A1 (0.32) IDO1
SCHEMBL6960778 0.83 LMNA (0.34) IDO1GRM2NAMPTKMT2ACYP3A4
SCHEMBL6972999 0.83 RXFP1 (0.37) KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed