SCHEMBL6967430

SCHEMBL6967430

CC(=O)OC(Cc1cccnc1)c1nc(C(C)C)c(Sc2cccc(Cl)c2)[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
LMNA P02545 1/20 0.41
IDO1 P14902 2/20 0.36
NPC1 O15118 4/20 0.35
GRM5 P41594 1/20 0.34
KDM4E B2RXH2 1/20 0.33
USP2 O75604 1/20 0.33
ALOX15 P16050 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RAB9A P51151 2/20 0.33
RORC P51449 1/20 0.33
CSNK2A2 P19784 1/20 0.33
CSNK2B P67870 1/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP51A1 Q16850 1/20 0.33
PLA2G7 Q13093 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973278 0.93 MEN1 (0.35) ALDH1A1LMNAIDO1NPC1KDM4E
SCHEMBL7081545 0.90 CSNK2A2 (0.34) ALDH1A1LMNAKDM4ECSNK2A2CSNK2B
SCHEMBL7084647 0.90 ALDH1A1 (0.38) ALDH1A1LMNAIDO1NPC1GRM5
SCHEMBL6972343 0.90 IDO1 (0.36) ALDH1A1LMNAIDO1KDM4ERORC
SCHEMBL6969311 0.89 LMNA (0.37) LMNAIDO1KDM4EKMT2ASMN1; SMN2
SCHEMBL6972366 0.87 ALDH1A1 (0.37) ALDH1A1LMNAIDO1NPC1GRM5
SCHEMBL6972999 0.87 RXFP1 (0.37) ALDH1A1LMNAKDM4ENPSR1RAB9A
SCHEMBL6970038 0.86 ALDH1A1 (0.41) ALDH1A1LMNAIDO1NPC1KDM4E
SCHEMBL7079754 0.86 IDO1 (0.37) IDO1KDM4ERORCKMT2A
SCHEMBL7081642 0.85 TP53 (0.39) LMNAGRM5MEN1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed