SCHEMBL6974922

SCHEMBL6974922

CC(C)c1nc(CN(C)C)n(Cc2cccnc2)c1Sc1cccc(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.41
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
ALDH1A1 P00352 3/20 0.37
LMNA P02545 2/20 0.37
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
P2RX7 Q99572 1/20 0.36
GABRA5 P31644 2/20 0.35
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GABRA1 P14867 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967631 0.93 CHRNB2 (0.39) POLBCHRNB2CHRNA4LMNAGRIN1
SCHEMBL6963923 0.91 POLB (0.44) POLBSLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL7079895 0.89 GRIN1 (0.38) CHRNB2CHRNA4GRIN1GRIN2BTSHR
SCHEMBL6965787 0.89 ALDH1A1 (0.38) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6970034 0.89 ALDH1A1 (0.40) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL7085922 0.88 CHRNB2 (0.42) CHRNB2CHRNA4ALDH1A1LMNAGABRA5
SCHEMBL7085996 0.87 ALDH1A1 (0.39) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6971118 0.87 ALDH1A1 (0.37) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6965333 0.87 ALDH1A1 (0.41) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6974920 0.86 ALDH1A1 (0.37) ALDH1A1LMNAGRIN1GRIN2BP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed