SCHEMBL708062

SCHEMBL708062

COc1cccc(NC=C2C(=O)OC(C)(C)OC2=O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 16/20 1.00
HSD17B10 Q99714 4/20 1.00
MAPK1 P28482 1/20 1.00
CYP1A2 P05177 2/20 0.66
CYP3A4 P08684 2/20 0.66
CASP1 P29466 2/20 0.64
CASP7 P55210 2/20 0.64
RAB9A P51151 1/20 0.61
TSHR P16473 1/20 0.58
L3MBTL1 Q9Y468 2/20 0.51
NPSR1 Q6W5P4 2/20 0.48
KDM4E B2RXH2 1/20 0.48
HPGD P15428 1/20 0.48
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
POLB P06746 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015141 1.00 ALDH1A1 (1.00) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL19850580 0.88 ALDH1A1 (0.79) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL2209335 0.87 ALDH1A1 (0.76) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL3059418 0.84 ALDH1A1 (0.72) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL16134952 0.82 ALDH1A1 (0.69) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL12003807 0.81 ALDH1A1 (0.67) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL25544341 0.81 ALDH1A1 (0.71) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL12830164 0.81 ALDH1A1 (0.67) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL2209684 0.81 ALDH1A1 (0.67) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL374339 0.80 ALDH1A1 (0.67) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115368301-B Preparation method of 4-hydroxy-7-methoxyquinoline 常州琦诺生物科技有限公司 2023-10-20 CN claimed
CN-115368301-A Preparation method of 4-hydroxy-7-methoxyquinoline 常州琦诺生物科技有限公司 2022-11-22 CN claimed
CN-115368301-B Preparation method of 4-hydroxy-7-methoxyquinoline 常州琦诺生物科技有限公司 2023-10-20 CN disclosed
CN-115368301-A Preparation method of 4-hydroxy-7-methoxyquinoline 常州琦诺生物科技有限公司 2022-11-22 CN disclosed
US-9957233-B1 Process for preparing substituted quinolin-4-ol compounds CALITOR SCIENCES, LLC (US) 2018-05-01 US disclosed
US-9957233-B1 Process for preparing substituted quinolin-4-ol compounds CALITOR SCIENCES, LLC (US) 2018-05-01 US disclosed
WO-2018026877-A1 PROCESS FOR PREPARING SUBSTITUTED QUINOLIN-4-OL COMPOUNDS CALITOR SCIENCES, LLC (US) 2018-02-08 WO disclosed
WO-2018026877-A1 PROCESS FOR PREPARING SUBSTITUTED QUINOLIN-4-OL COMPOUNDS CALITOR SCIENCES, LLC (US) 2018-02-08 WO disclosed
US-9636375-B2 Hepatitis C virus inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2017-05-02 US disclosed
US-9636375-B2 Hepatitis C virus inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2017-05-02 US disclosed
US-20160067302-A1 Hepatitis C Virus Inhibitors BRISTOL MYERS SQUIBB CO (US) 2016-03-10 US disclosed
US-6867185-B2 Inhibitors of hepatitis C virus BRISTOL-MYERS SQUIBB COMPANY (US) 2005-03-15 US disclosed
EP-1505963-A1 HEPATITIS C VIRUS INHIBITORS Bristol-Myers Squibb Company (US) 2005-02-16 EP disclosed
EP-1455809-A2 INHIBITORS OF HEPATITIS C VIRUS Bristol-Myers Squibb Company (US) 2004-09-15 EP disclosed
US-20040106559-A1 Hepatitis C virus inhibitors BRISTOL-MYERS SQUIBB COMPANY 2004-06-03 US disclosed
US-20040038872-A1 Inhibitors of hepatitis C virus BRISTOL-MYERS SQUIBB COMPANY 2004-02-26 US disclosed
WO-2003099274-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-12-04 WO disclosed
WO-2003099274-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-12-04 WO disclosed
WO-2003053349-A2 INHIBITORS OF HEPATITIS C VIRUS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-07-03 WO disclosed
WO-2003053349-A2 INHIBITORS OF HEPATITIS C VIRUS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-07-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160067302-A1 Hepatitis C Virus Inhibitors HAVCR2, HCCS, CTRB1 ALDH1A1 769/4885HSD17B10 553/4885MAPK1 2557/4885
US-20040038872-A1 Inhibitors of hepatitis C virus HAVCR2, LIPC, ZC3HAV1 ALDH1A1 576/4885HSD17B10 1615/4885MAPK1 2287/4885
US-20040106559-A1 Hepatitis C virus inhibitors HAVCR2, HCCS, RNASE1 ALDH1A1 512/4885HSD17B10 735/4885MAPK1 1573/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.