Quinoline

Quinoline

SCHEMBL7081987

CC(N)C(=O)O.c1ccc2ncccc2c1

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.59
NPSR1 Q6W5P4 2/20 0.46
RXFP1 Q9HBX9 2/20 0.46
KDM4E B2RXH2 2/20 0.46
PRNP P04156 1/20 0.46
MAPK10 P53779 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
LMNA P02545 1/20 0.45
AKR1C3 P42330 1/20 0.44
AKR1C2 P52895 1/20 0.44
PABPC1 P11940 1/20 0.43
ELANE P08246 1/20 0.43
ALOX15 P16050 1/20 0.43
HTT P42858 1/20 0.43
PLK1 P53350 1/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL7081988 1.00 ALDH1A1 (0.59) ALDH1A1NPSR1RXFP1KDM4EPRNP
Quinoline SCHEMBL4747553 0.90 ALDH1A1 (0.55) ALDH1A1NPSR1RXFP1KDM4EPRNP
Quinoline SCHEMBL5874361 0.88 ALDH1A1 (0.61) ALDH1A1NPSR1RXFP1KDM4EPRNP
Quinoline SCHEMBL27820159 0.88 ALDH1A1 (0.61) ALDH1A1NPSR1RXFP1KDM4EPRNP
Quinoline SCHEMBL5874375 0.88 ALDH1A1 (0.61) ALDH1A1NPSR1RXFP1KDM4EPRNP
Oxyquinoline SCHEMBL28087250 0.87 ALDH1A1 (0.57) ALDH1A1KDM4ESMN1; SMN2LMNAMEN1
Quinoline SCHEMBL4265433 0.85 ALDH1A1 (0.68) ALDH1A1KDM4ESMN1; SMN2LMNAALOX15
Quinoxaline SCHEMBL28009513 0.85 NPSR1 (0.46) ALDH1A1NPSR1RXFP1KDM4EPRNP
Quinoline SCHEMBL5272119 0.85 ALDH1A1 (0.74) ALDH1A1KDM4ESMN1; SMN2PABPC1ALOX15
Quinoline SCHEMBL2201840 0.85 ALDH1A1 (0.74) ALDH1A1KDM4ESMN1; SMN2PABPC1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106047846-A An 8-hydroxyquinoline alanine translation system and applications thereof 中国科学院生物物理研究所 2016-10-26 CN claimed
CN-104059891-B 8-hydroxyquinoline alanine translation system and application thereof 中国科学院生物物理研究所 2016-08-17 CN claimed
US-20220168383-A1 NEUROTENSINERGIC AGONISTS AND METHODS OF USING SAME PREVENTING OR TREATING PAIN SOCPRA SCIENCES SANTÉ ET HUMAINES S.E.C. (CA) 2022-06-02 US disclosed
EP-3921331-A1 NEUROTENSINERGIC AGONISTS AND METHODS OF USING SAME PREVENTING OR TREATING PAIN Socpra Sciences Santé Et Humaines S.E.C. (CA) 2021-12-15 EP disclosed
WO-2020160685-A1 NEUROTENSINERGIC AGONISTS AND METHODS OF USING SAME PREVENTING OR TREATING PAIN SOCPRA Sciences Sante et Humaines S.E.C. (CA) 2020-08-13 WO disclosed
CN-103122024-B AntiHIV1 RT activity infection polypeptide, composition and the purposes of engineer 中国人民解放军军事医学科学院毒物药物研究所 2017-12-29 CN disclosed
CN-106047846-A An 8-hydroxyquinoline alanine translation system and applications thereof 中国科学院生物物理研究所 2016-10-26 CN disclosed
CN-104059891-B 8-hydroxyquinoline alanine translation system and application thereof 中国科学院生物物理研究所 2016-08-17 CN disclosed
EP-1322616-A2 QUINOLINE-(C=O)-(DI-, TRI- AND TETRAPEPTIDE) DERIVATIVES AS CASPASE INHIBITORS ENZYME SYSTEMS PRODUCTS INC. (US) 2003-07-02 EP disclosed
WO-2002018341-A9 QUINOLINE- (C=O) - (DI-, TRI- AND TETRAPEPTIDE) DERIVATIVES AS CASPASE INHIBITORS ENZYME SYST PROD INC (US) 2002-11-21 WO disclosed
US-20020052323-A1 Quinoline-(C=O)-(multiple amino acids)-leaving group compounds for pharmaceutical compositions and reagents MP BIOMEDICALS, LLC 2002-05-02 US disclosed
WO-2002018341-A2 QUINOLINE- (C=O) - (DI-, TRI- AND TETRAPEPTIDE) DERIVATIVES AS CASPASE INHIBITORS ENZYME SYSTEMS PRODUCTS, INC. (US) 2002-03-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220168383-A1 NEUROTENSINERGIC AGONISTS AND METHODS OF USING SAME PREVENTING OR TREATING PAIN VIP, NTSR2, VIPR2 ALDH1A1 1872/4885NPSR1 17/4885RXFP1 23/4885
US-20020052323-A1 Quinoline-(C=O)-(multiple amino acids)-leaving group compounds for pharmaceutical compositions and reagents CASP3, CASP1, BAX ALDH1A1 1648/4885NPSR1 3170/4885RXFP1 1482/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.