SCHEMBL7082250

SCHEMBL7082250

CC(C)(C)OC(=O)Nc1ccc(NC(=O)c2ccnc3ccccc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.51
NR2E1 Q9Y466 3/20 0.49
DNMT1 P26358 2/20 0.48
DNMT3A Q9Y6K1 2/20 0.48
DNMT3L Q9UJW3 1/20 0.48
MAP4K4 O95819 1/20 0.47
RORA P35398 1/20 0.47
ABCB1 P08183 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.46
CYP3A4 P08684 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CYP1A2 P05177 1/20 0.46
GAA P10253 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
NR4A1 P22736 1/20 0.46
ESR2 Q92731 1/20 0.46
ACLY P53396 1/20 0.46
KDR P35968 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29406849 0.84 MEN1 (0.53) NR2E1RORAMEN1KMT2AGAA
SCHEMBL379808 0.81 CYP3A4 (0.60) NR2E1DNMT1DNMT3ADNMT3LCYP3A4
SCHEMBL804472 0.80 CYP3A4 (0.50) NR2E1DNMT1DNMT3ADNMT3LRORA
SCHEMBL6815971 0.80 NPC1 (0.66) NAMPTMEN1KMT2AL3MBTL1
SCHEMBL17981164 0.79 PTPN1 (0.56) DNMT1DNMT3ADNMT3LMAP4K4MEN1
SCHEMBL7784318 0.79 DNMT1 (0.65) NR2E1DNMT1DNMT3ADNMT3LRORA
SCHEMBL6811232 0.78 FLT3 (0.58) NAMPTMAP4K4MEN1KMT2AGAA
SCHEMBL28176881 0.77 LMNA (0.45) ABCB1ABCG2CYP3A4MEN1KMT2A
SCHEMBL6814808 0.77 SMN1; SMN2 (0.63) NAMPTKDRHTT
SCHEMBL8088287 0.76 CYP17A1 (0.46) NAMPTDNMT1DNMT3AMAP4K4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030036653-A1 Diaminopyridine-containing thiourea inhibitors of herpes viruses AMERICAN HOME PRODUCTS CORPORATION 2003-02-20 US disclosed
US-6410571-B1 VIRICIDES AMERICAN HOME PRODUCTS CORPORATION 2002-06-25 US disclosed
US-20020026055-A1 Aminopyridine-containing thiourea inhibitors of herpes viruses AMERICAN HOME PRODUCTS CORPORATION 2002-02-28 US disclosed
US-20010039348-A1 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group AMERICAN HOME PRODUCTS CORPORATION (US) 2001-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030036653-A1 Diaminopyridine-containing thiourea inhibitors of herpes viruses HAVCR2, CCR6, CXCR6 NAMPT 3260/4885NR2E1 600/4885DNMT1 1647/4885
US-20010039348-A1 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group CCR6, HAVCR2, BCOR NAMPT 3999/4885NR2E1 266/4885DNMT1 1206/4885
US-20020026055-A1 Aminopyridine-containing thiourea inhibitors of herpes viruses TK1, TPMT, CXCR6 NAMPT 4031/4885NR2E1 1125/4885DNMT1 2257/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.