SCHEMBL7082472

SCHEMBL7082472

CC(C)c1nc(CCO)n(Cc2ccccn2)c1Sc1cccc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
KMT2A Q03164 4/20 0.37
MAPT P10636 3/20 0.37
PPP1CA P62136 1/20 0.37
GRM5 P41594 1/20 0.36
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
KDM4E B2RXH2 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
PKM P14618 1/20 0.35
TP53 P04637 2/20 0.34
MEN1 O00255 3/20 0.33
HPGD P15428 2/20 0.33
AGTR1 P30556 1/20 0.33
HRH1 P35367 1/20 0.33
THRB P10828 1/20 0.33
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974023 0.94 TLR8 (0.36) ALDH1A1KMT2AMAPTPPP1CAGRM5
SCHEMBL7082531 0.92 HRH1 (0.34) ALDH1A1KMT2AMAPTGRIN1GRIN2B
SCHEMBL7079929 0.92 GRM5 (0.38) ALDH1A1KMT2AMAPTPPP1CAGRM5
SCHEMBL6967528 0.91 GRM5 (0.36) ALDH1A1KMT2AMAPTPPP1CAGRM5
SCHEMBL7084157 0.89 TLR7 (0.37) ALDH1A1KDM4ETP53HRH1LMNA
SCHEMBL8507295 0.89 HRH3 (0.39) ALDH1A1KMT2AMAPTPPP1CAGRM5
SCHEMBL6973313 0.89 GRIN1 (0.38) ALDH1A1KMT2AMAPTGRIN1GRIN2B
SCHEMBL6962202 0.89 GRM5 (0.38) ALDH1A1KMT2AMAPTPPP1CAGRM5
SCHEMBL6960270 0.88 ALDH1A1 (0.36) ALDH1A1KMT2AMAPTPPP1CAGRM5
SCHEMBL6973417 0.87 MAPT (0.37) ALDH1A1KMT2AMAPTPPP1CAGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed