SCHEMBL7083459

SCHEMBL7083459

CC(C)c1nc(COCCOC(N)=O)n(Cc2cccnc2)c1Sc1cccc(F)c1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 7/20 0.35
GRIN2B Q13224 7/20 0.35
S1PR3 Q99500 4/20 0.33
PTAFR P25105 2/20 0.32
GRM2 Q14416 1/20 0.32
IDO1 P14902 1/20 0.32
LMNA P02545 1/20 0.32
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
GFER P55789 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973065 0.94 GRIN1 (0.35) GRIN1GRIN2BS1PR3GRM2IDO1
SCHEMBL6960775 0.93 GRIN1 (0.35) GRIN1GRIN2BS1PR3PTAFRIDO1
SCHEMBL7080841 0.93 GRIN1 (0.36) GRIN1GRIN2BS1PR3PTAFRGRM2
SCHEMBL6969763 0.92 GRIN1 (0.35) GRIN1GRIN2BS1PR3PTAFRGRM2
SCHEMBL7082343 0.91 GRIN1 (0.32) GRIN1GRIN2BLMNAMAPT
SCHEMBL6969475 0.91 ALDH1A1 (0.37) GRIN1GRIN2BS1PR3GRM2LMNA
SCHEMBL6960297 0.90 MDM2 (0.34) S1PR3LMNAALDH1A1KMT2A
SCHEMBL6962104 0.89 GRIN1 (0.36) GRIN1GRIN2BS1PR3
SCHEMBL6972478 0.89 RXFP1 (0.38) LMNAALDH1A1MAPT
SCHEMBL6973962 0.88 ADRA1D (0.35) S1PR3ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed