SCHEMBL6973065

SCHEMBL6973065

CC(C)c1nc(COCCOC(N)=O)n(Cc2cccnc2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.35
GRIN2B Q13224 2/20 0.35
S1PR3 Q99500 4/20 0.34
GRM2 Q14416 2/20 0.33
TLR7 Q9NYK1 4/20 0.33
IDO1 P14902 1/20 0.33
SCN9A Q15858 1/20 0.32
ENPP2 Q13822 1/20 0.32
PKM P14618 1/20 0.31
RORC P51449 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7083459 0.94 GRIN1 (0.35) GRIN1GRIN2BS1PR3GRM2IDO1
SCHEMBL7082204 0.93 GRIN1 (0.35) GRIN1GRIN2BS1PR3TLR7IDO1
SCHEMBL6974966 0.93 GRIN1 (0.36) GRIN1GRIN2BS1PR3GRM2TLR7
SCHEMBL6967126 0.93 GRIN1 (0.37) GRIN1GRIN2BS1PR3GRM2TLR7
SCHEMBL6970826 0.91 GRIN1 (0.35) GRIN1GRIN2BS1PR3GRM2TLR7
SCHEMBL6973962 0.91 ADRA1D (0.35) S1PR3TLR7PKM
SCHEMBL6960297 0.90 MDM2 (0.34) S1PR3TLR7
SCHEMBL6961792 0.90 ENPP2 (0.32) ENPP2
SCHEMBL6973898 0.88 GRIN1 (0.35) GRIN1GRIN2BS1PR3TLR7IDO1
SCHEMBL6969475 0.88 ALDH1A1 (0.37) GRIN1GRIN2BS1PR3GRM2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed