SCHEMBL6973962

SCHEMBL6973962

CC(C)c1nc(COCCOC(N)=O)n(Cc2cccnc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 1/20 0.35
SLC16A3 O15427 1/20 0.33
TLR7 Q9NYK1 3/20 0.33
GABRA1 P14867 2/20 0.33
GABRA5 P31644 2/20 0.33
S1PR3 Q99500 2/20 0.32
KMT2A Q03164 2/20 0.32
CACNA1I Q9P0X4 1/20 0.32
GRM5 P41594 1/20 0.32
PKM P14618 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90B1 P14625 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MCL1 Q07820 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969475 0.94 ALDH1A1 (0.37) ADRA1DSLC16A3GABRA1GABRA5S1PR3
SCHEMBL6969211 0.93 KMT2A (0.34) SLC16A3GABRA1GABRA5S1PR3KMT2A
SCHEMBL6966178 0.93 ADRA1D (0.36) ADRA1DGABRA1GABRA5S1PR3KMT2A
SCHEMBL6957033 0.93 ADRA1D (0.37) ADRA1DSLC16A3TLR7GABRA1GABRA5
SCHEMBL6966597 0.91 FKBP1A (0.35) ADRA1DTLR7GABRA1GABRA5S1PR3
SCHEMBL6961932 0.91 PIM1 (0.33) KMT2AMEN1
SCHEMBL6973065 0.91 GRIN1 (0.35) TLR7S1PR3PKM
SCHEMBL6960297 0.90 MDM2 (0.34) TLR7GABRA1GABRA5S1PR3KMT2A
SCHEMBL7085225 0.88 GRM5 (0.33) SLC16A3TLR7GABRA1GABRA5S1PR3
SCHEMBL7083459 0.88 GRIN1 (0.35) S1PR3KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed