SCHEMBL7083557

SCHEMBL7083557

COc1cc(C=CC=C2SC(O)NC2O)ccc1OC(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 4/20 0.39
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HDAC1 Q13547 2/20 0.38
HDAC2 Q92769 2/20 0.38
HDAC8 Q9BY41 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4A P27815 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
TRPA1 O75762 1/20 0.37
MTNR1A P48039 1/20 0.37
ALDH1A1 P00352 2/20 0.36
APP P05067 1/20 0.36
CYP1B1 Q16678 3/20 0.35
CYP1A2 P05177 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7083561 1.00 CYP1A1 (0.39) CYP1A1PTGS1PTGS2MEN1KMT2A
SCHEMBL7083564 0.72 DNMT1 (0.39) CYP1A1PTGS1PTGS2MEN1KMT2A
SCHEMBL6966722 0.71 XDH (0.60) CYP1A1PTGS1PTGS2MEN1KMT2A
SCHEMBL6966726 0.71 XDH (0.60) CYP1A1PTGS1PTGS2MEN1KMT2A
SCHEMBL8335512 0.70 PDE4B (0.46) MEN1KMT2AHDAC1HDAC2HDAC8
SCHEMBL6972866 0.70 PDE4B (0.58) MEN1KMT2APDE4BALDH1A1HPGD
SCHEMBL6972871 0.70 PDE4B (0.58) MEN1KMT2APDE4BALDH1A1HPGD
SCHEMBL29096342 0.68 KDM4E (0.57) MEN1KMT2AHDAC1HDAC2HDAC8
SCHEMBL16960211 0.68 ALDH1A1 (0.47) CYP1A1PTGS1PTGS2MEN1KMT2A
SCHEMBL6587547 0.68 MMP9 (0.58) CYP1A1PTGS1PTGS2HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0783496-B9 THIAZOLIDINEDIONE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-09-03 EP disclosed
EP-0783496-B1 THIAZOLIDINEDIONE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-26 EP disclosed