SCHEMBL7084539

SCHEMBL7084539

CCC(OCCOC(C)=O)c1nc(C(C)C)c(Sc2cccc(F)c2)[nH]1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 5/20 0.33
GCGR P47871 1/20 0.31
TYMS P04818 1/20 0.31
CA2 P00918 1/20 0.30
CA4 P22748 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7082473 0.90 SLC6A9 (0.34) SLC6A9GCGRTYMSCA2CA4
SCHEMBL7086458 0.89 TP53 (0.36) SLC6A9TYMSLMNA
SCHEMBL7086334 0.89 DHFR (0.32) CA2CA4ALDH1A1L3MBTL1
SCHEMBL7086009 0.88 SLC6A9 (0.30) SLC6A9
SCHEMBL6974498 0.88 SLC6A9 (0.35) SLC6A9GCGRTYMSCA2CA4
SCHEMBL7081199 0.88 SLC6A9 (0.33) SLC6A9GCGRTYMS
SCHEMBL7078551 0.87 SLC6A9 (0.33) SLC6A9
SCHEMBL6971934 0.86 CACNA1C (0.35) LMNA
SCHEMBL6960778 0.86 LMNA (0.34) ALDH1A1LMNA
SCHEMBL6966214 0.83

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed