SCHEMBL6973819

SCHEMBL6973819

CCn1c(CNS(C)(=O)=O)nc(C(C)C)c1Sc1cccc(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
LMNA P02545 2/20 0.34
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
S1PR1 P21453 3/20 0.33
TYMS P04818 2/20 0.33
HPGD P15428 1/20 0.33
TDP1 Q9NUW8 2/20 0.32
GRM5 P41594 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974402 0.90 TDP1 (0.32) S1PR1TDP1
SCHEMBL6973826 0.88 ALDH1A1 (0.34) LMNATYMSNPSR1
SCHEMBL6968203 0.88 MAOB (0.36) TP53RXFP1ADRB2ADRB1ADRB3
SCHEMBL6972096 0.88 LMNA (0.37) TP53RXFP1LMNAADRB2ADRB1
SCHEMBL7084653 0.87 SETDB1 (0.33) TSHR
SCHEMBL7080431 0.86 MEN1 (0.36) TP53RXFP1LMNATYMSHPGD
SCHEMBL7086513 0.85 GRIN1 (0.36) TP53LMNAHPGDGRM5KMT2A
SCHEMBL6975217 0.85 TP53 (0.39) TP53RXFP1LMNAADRB2ADRB1
SCHEMBL7084297 0.85 LMNA (0.40) TP53LMNATDP1KMT2A
SCHEMBL7088075 0.85 MAPT (0.37) LMNAHPGDMEN1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed