SCHEMBL7085225

SCHEMBL7085225

CC(C)c1nc(COCCO)n(Cc2cccnc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.33
SRC P12931 1/20 0.33
GABRA5 P31644 3/20 0.33
GABRA1 P14867 2/20 0.33
HIF1A Q16665 1/20 0.32
SLC16A3 O15427 1/20 0.32
TLR7 Q9NYK1 3/20 0.32
S1PR3 Q99500 1/20 0.32
KMT2A Q03164 2/20 0.31
CACNA1I Q9P0X4 1/20 0.31
PKM P14618 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TP53 P04637 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972360 0.93 ALDH1A1 (0.37) GRM5SRCGABRA5GABRA1HIF1A
SCHEMBL6970649 0.90 KCNH2 (0.32) GRM5
SCHEMBL6973898 0.90 GRIN1 (0.35) SRCTLR7S1PR3PKM
SCHEMBL6969211 0.89 KMT2A (0.34) GRM5GABRA5GABRA1HIF1ASLC16A3
SCHEMBL7085466 0.89 ALOX5AP (0.34) SRCHIF1ATLR7KMT2AALDH1A1
SCHEMBL6973962 0.88 ADRA1D (0.35) GRM5GABRA5GABRA1SLC16A3TLR7
SCHEMBL7087528 0.88 SRC (0.35) SRCGABRA5GABRA1HIF1ATLR7
SCHEMBL6973652 0.88 SRC (0.37) SRCGABRA5GABRA1TLR7KMT2A
SCHEMBL6969270 0.86 TLR7 (0.35) SRCGABRA5GABRA1TLR7KMT2A
SCHEMBL6962104 0.86 GRIN1 (0.36) SRCTLR7S1PR3PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed