SCHEMBL7087918

SCHEMBL7087918

Oc1cc(Cl)c(Oc2ccc3[nH]cc(CC4CCCCC4)c3c2)c(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.42
HTR1B P28222 3/20 0.42
HTR1D P28221 1/20 0.42
HTR6 P50406 1/20 0.40
THRA P10827 6/20 0.40
THRB P10828 6/20 0.40
SLC6A4 P31645 2/20 0.38
S1PR1 P21453 1/20 0.38
BCHE P06276 2/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6516005 0.86 THRB (0.56) HTR1AHTR1BHTR1DTHRATHRB
SCHEMBL7090308 0.86 THRA (0.41) HTR1AHTR1BHTR1DHTR6THRA
SCHEMBL6513360 0.85 THRB (0.45) HTR1AHTR1BHTR1DHTR6THRA
SCHEMBL6518665 0.85 THRB (0.57) THRATHRBS1PR1
SCHEMBL6519233 0.84 THRA (0.46) HTR1AHTR1BHTR1DTHRATHRB
SCHEMBL7088286 0.84 HTR1A (0.41) HTR1AHTR1BHTR1DHTR6THRA
SCHEMBL6519539 0.83 THRA (0.48) HTR1AHTR1BHTR1DHTR6THRA
SCHEMBL7090048 0.83 THRA (0.41) HTR1AHTR1BHTR1DHTR6THRA
SCHEMBL7085216 0.83 THRA (0.44) HTR1AHTR1BHTR6THRATHRB
SCHEMBL7086371 0.83 HTR1A (0.48) HTR1AHTR1BHTR1DHTR6THRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347959-A1 INDOLE DERIVATIVES AS LIGANDS OF THYROID RECEPTORS Bayer Aktiengesellschaft (DE) 2003-10-01 EP disclosed
WO-2002051805-A1 INDOLE DERIVATIVES AS LIGANDS OF THYROID RECEPTORS BAYER AKTIENGESELLSCHAFT (DE) 2002-07-04 WO disclosed